SCHEMBL7417299

SCHEMBL7417299

CCOC(=O)/C(C)=C/c1cccc(C#N)c1

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDCD1 Q15116 1/20 0.74
CD274 Q9NZQ7 1/20 0.74
MAPT P10636 3/20 0.53
KMT2A Q03164 4/20 0.49
ALDH1A1 P00352 4/20 0.49
LMNA P02545 2/20 0.49
KDM4E B2RXH2 1/20 0.49
FBP1 P09467 2/20 0.49
MEN1 O00255 3/20 0.47
CYP1A2 P05177 1/20 0.46
GRM5 P41594 1/20 0.46
GLO1 Q04760 1/20 0.45
PKM P14618 1/20 0.44
HTT P42858 1/20 0.44
S1PR4 O95977 1/20 0.43
S1PR1 P21453 1/20 0.43
MAPK1 P28482 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
P4HB P07237 2/20 0.43
PTP4A1 Q93096 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10375509 0.87 PDCD1 (0.71) PDCD1CD274MAPTKMT2AALDH1A1
SCHEMBL10848993 0.87 PDCD1 (0.71) PDCD1CD274MAPTKMT2AALDH1A1
SCHEMBL21457292 0.85 PDCD1 (1.00) PDCD1CD274MAPTKMT2AALDH1A1
SCHEMBL21457289 0.85 PDCD1 (1.00) PDCD1CD274MAPTKMT2AALDH1A1
SCHEMBL20786827 0.83 MAPT (0.51) PDCD1CD274MAPTKMT2AALDH1A1
SCHEMBL20787944 0.83 MAPT (0.51) PDCD1CD274MAPTKMT2AALDH1A1
SCHEMBL14113061 0.81 KMT2A (0.53) PDCD1CD274MAPTKMT2AALDH1A1
SCHEMBL21065588 0.81 KMT2A (0.53) PDCD1CD274MAPTKMT2AALDH1A1
SCHEMBL3115027 0.81 AKR1C3 (0.59) PDCD1CD274KDM4EFBP1P4HB
SCHEMBL6981746 0.81 AKR1C3 (0.59) PDCD1CD274KDM4EFBP1P4HB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0934265-A1 AMIDINOPHENYL-PYRROLIDINES, -PYRROLINES, AND -ISOXAZOLIDINES AND DERIVATIVES THEREOF Du Pont Pharmaceuticals Company (US) 1999-08-11 EP disclosed
WO-1998006694-A1 AMIDINOPHENYL-PYRROLIDINES, -PYRROLINES, AND -ISOXAZOLIDINES AND DERIVATIVES THEREOF DU PONT PHARMACEUTICALS COMPANY (US) 1998-02-19 WO disclosed