SCHEMBL7417401

SCHEMBL7417401

CCCc1cc(C)cc(C(Nc2ccc(C(=N)NO)cc2)C(=O)O)c1OCCO

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
F10 P00742 14/20 0.41
F7 P08709 14/20 0.41
F3 P13726 13/20 0.41
PRSS1 P07477 13/20 0.41
PRSS2 P07478 12/20 0.41
PRSS3 P35030 12/20 0.41
F2 P00734 11/20 0.39
CYP2C9 P11712 2/20 0.35
IDO1 P14902 2/20 0.35
KCNH2 Q12809 1/20 0.33
PPARG P37231 3/20 0.32
PPARA Q07869 3/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5883570 0.90 F7 (0.52) F10F7F3PRSS1PRSS2
SCHEMBL5883607 0.83 CYP2C9 (0.35) F10F7F3PRSS1PRSS2
SCHEMBL5882844 0.82 F7 (0.45) F10F7F3PRSS1PRSS2
SCHEMBL5883206 0.80 F10 (0.38) F10F7F3PRSS1PRSS2
SCHEMBL5883155 0.80 F7 (0.41) F10F7F3PRSS1PRSS2
SCHEMBL5883527 0.80 F7 (0.52) F10F7F3PRSS1PRSS2
Hydrochloric Acid SCHEMBL5883090 0.79 F7 (0.51) F10F7F3PRSS1PRSS2
SCHEMBL5882190 0.79 F10 (0.50) F10F7F3PRSS1PRSS2
SCHEMBL5883062 0.79 F7 (0.47) F10F7F3PRSS1PRSS2
SCHEMBL5882615 0.78 F10 (0.39) F10F7F3PRSS1PRSS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1149069-A1 PHENYLGLYCINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2001-10-31 EP disclosed
WO-2000035858-A1 PHENYLGLYCINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2000-06-22 WO disclosed