SCHEMBL741802

SCHEMBL741802

COCCCn1c(C2CCCN(C(=O)CC(N)Cc3ccc(-c4cccnc4)cc3)C2)nc2ccccc21

nearest known ligand 0.42

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 11/20 0.42
CYP2D6 P10635 7/20 0.42
KCNH2 Q12809 11/20 0.41
CHRM1 P11229 3/20 0.41
CYP3A4 P08684 1/20 0.38
ITK Q08881 1/20 0.38
PROKR1 Q8TCW9 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL740944 1.00 HRH1 (0.42) HRH1CYP2D6KCNH2CHRM1CYP3A4
SCHEMBL738739 0.94 HRH1 (0.46) HRH1CYP2D6KCNH2CHRM1CYP3A4
SCHEMBL738740 0.94 HRH1 (0.46) HRH1CYP2D6KCNH2CHRM1CYP3A4
SCHEMBL739066 0.93 HRH1 (0.42) HRH1CYP2D6KCNH2CHRM1CYP3A4
SCHEMBL739065 0.93 HRH1 (0.42) HRH1CYP2D6KCNH2CHRM1CYP3A4
SCHEMBL740155 0.93 HRH1 (0.45) HRH1CYP2D6KCNH2CHRM1CYP3A4
SCHEMBL740154 0.93 HRH1 (0.45) HRH1CYP2D6KCNH2CHRM1CYP3A4
SCHEMBL739975 0.92 DPP4 (0.45) HRH1CYP2D6KCNH2CHRM1CYP3A4
SCHEMBL739976 0.92 DPP4 (0.45) HRH1CYP2D6KCNH2CHRM1CYP3A4
SCHEMBL763510 0.92 HRH1 (0.43) HRH1CYP2D6KCNH2CHRM1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US claimed
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed