SCHEMBL7418280

SCHEMBL7418280

COC(=O)c1cccc(-n2c(=O)n(Cc3ccccc3)c(=O)c3[nH]cnc32)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 8/20 1.00
PDE4B Q07343 8/20 1.00
PDE4C Q08493 8/20 1.00
PDE4D Q08499 8/20 1.00
OPRK1 P41145 2/20 0.74
KMT2A Q03164 4/20 0.69
POLB P06746 2/20 0.60
MEN1 O00255 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7417624 0.85 PDE4A (1.00) PDE4APDE4BPDE4CPDE4DOPRK1
SCHEMBL7422131 0.83 PDE4A (0.71) PDE4APDE4BPDE4CPDE4DOPRK1
SCHEMBL7420809 0.83 PDE4A (1.00) PDE4APDE4BPDE4CPDE4DKMT2A
SCHEMBL2932520 0.83 PDE4A (0.70) PDE4APDE4BPDE4CPDE4DOPRK1
SCHEMBL6662589 0.82 PDE4A (1.00) PDE4APDE4BPDE4CPDE4DKMT2A
SCHEMBL7415138 0.82 PDE4A (1.00) PDE4APDE4BPDE4CPDE4DKMT2A
SCHEMBL8690835 0.81 PDE4A (0.80) PDE4APDE4BPDE4CPDE4DKMT2A
SCHEMBL8182797 0.81 PDE4A (0.80) PDE4APDE4BPDE4CPDE4DKMT2A
SCHEMBL1802317 0.81 PDE4A (0.68) PDE4APDE4BPDE4CPDE4DOPRK1
SCHEMBL7532671 0.81 PDE4A (0.76) PDE4APDE4BPDE4CPDE4DKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5821366-A Xanthines and their therapeutic use CHIROSCIENCE LIMITED (GB) 1998-10-13 US claimed
EP-0825993-A1 XANTHINES AND THEIR THERAPEUTIC USE Chiroscience Limited (GB) 1998-03-04 EP claimed
WO-1996036638-A1 XANTHINES AND THEIR THERAPEUTIC USE CHIROSCIENCE LIMITED (GB) 1996-11-21 WO claimed
US-5821366-A Xanthines and their therapeutic use CHIROSCIENCE LIMITED (GB) 1998-10-13 US disclosed