SCHEMBL7418341

SCHEMBL7418341

NCc1nc(Br)cnc1N

nearest known ligand 0.37

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.37
KMT2A Q03164 1/20 0.37
ATR Q13535 1/20 0.34
GRM5 P41594 1/20 0.32
NUDT1 P36639 1/20 0.32
MAPK1 P28482 1/20 0.31
MAPKAPK2 P49137 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14703937 0.82 HTT (0.37) HTTKMT2AATRGRM5MAPK1
SCHEMBL8055545 0.80 CCR4 (0.38) HTTKMT2AATRMAPKAPK2
SCHEMBL1585295 0.80 ATR (0.37) HTTKMT2AATRGRM5MAPK1
SCHEMBL30427027 0.80 CCR4 (0.38) HTTKMT2AATRMAPKAPK2
SCHEMBL25225301 0.78 CCR4 (0.32)
SCHEMBL30497655 0.78 CCR4 (0.32)
Hydrochloric Acid SCHEMBL30450382 0.77 CCR4 (0.31)
SCHEMBL27870217 0.77 HTT (0.33) HTTKMT2AATR
SCHEMBL20839003 0.77 ADORA2A (0.35) HTTKMT2AATR
Hydrochloric Acid SCHEMBL25225244 0.77 CCR4 (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5002944-A Compounds having cardiotonic activity RHONE-POULENC RORER PHARMACEUTICALS INC. (US) 1991-03-26 US disclosed
EP-0333727-A1 HETEROCYCLIC SUBSTITUTED BICYCLOUREAS HAVING CARDIOTONIC ACTIVITY RORER INTERNATIONAL (OVERSEAS) INC. (a Delaware corporation) (US) 1989-09-27 EP disclosed
US-4859672-A Pyrido[2,3-d]pyrimidinone and imidazo[4,5-b]pyrimidinone RORER PHARMACEUTICAL CORPORATION (US) 1989-08-22 US disclosed
WO-1988003025-A1 HETEROCYCLIC SUBSTITUTED BICYCLOUREAS HAVING CARDIOTONIC ACTIVITY RORER INTERNATIONAL (OVERSEAS) INC. (US) 1988-05-05 WO disclosed