SCHEMBL7419151

SCHEMBL7419151

CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)[C@@H]1C[C@@H](CCCC(F)(F)F)C(=O)O1

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ATM Q13315 1/20 0.41
SCN9A Q15858 5/20 0.40
CTSS P25774 2/20 0.40
CTSL P07711 1/20 0.40
CTSB P07858 1/20 0.40
CTSK P43235 1/20 0.40
ACE P12821 1/20 0.39
AKT1 P31749 1/20 0.38
REN P00797 1/20 0.38
ALDH1A1 P00352 1/20 0.37
APP P05067 1/20 0.37
PSMB5 P28074 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6836252 0.89 ATM (0.43) ATMSCN9ACTSSCTSLCTSB
SCHEMBL7397628 0.88 ATM (0.44) ATMSCN9ACTSSCTSLCTSB
SCHEMBL8270815 0.87 ATM (0.43) ATMSCN9ACTSSCTSLCTSB
SCHEMBL9473183 0.86 ATM (0.40) ATMSCN9ACTSSCTSLCTSB
SCHEMBL9831090 0.86 ATM (0.40) ATMSCN9ACTSSCTSLCTSB
SCHEMBL7584316 0.86 ATM (0.43) ATMCTSSCTSLCTSBCTSK
SCHEMBL7432732 0.86 ATM (0.46) ATMSCN9ACTSSCTSLCTSB
SCHEMBL9005035 0.86 ATM (0.46) ATMSCN9ACTSSCTSLCTSB
SCHEMBL6312228 0.86 ATM (0.46) ATMSCN9ACTSSCTSLCTSB
SCHEMBL7443701 0.86 ATM (0.46) ATMSCN9ACTSSCTSLCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5733882-A Retroviral protease inhibitors SMITHKLINE BEECHAM CORPORATION (US) 1998-03-31 US disclosed
EP-0602069-A4 RETROVIRAL PROTEASE INHIBITORS. SMITHKLINE BEECHAM CORP (US) 1995-05-03 EP disclosed
EP-0602069-A1 RETROVIRAL PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 1994-06-22 EP disclosed
WO-1993002057-A1 RETROVIRAL PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 1993-02-04 WO disclosed