SCHEMBL7419637

SCHEMBL7419637

N#Cc1cccc(CN2CCCC[C@H](N)C2=O)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIRT2 Q8IXJ6 1/20 0.46
SIRT1 Q96EB6 1/20 0.46
EPHX1 P07099 1/20 0.43
ROCK2 O75116 1/20 0.43
ROCK1 Q13464 1/20 0.43
DPP4 P27487 3/20 0.43
DPP7 Q9UHL4 2/20 0.43
FNTA P49354 1/20 0.43
FNTB P49356 1/20 0.43
HCRTR1 O43613 1/20 0.43
HCRTR2 O43614 1/20 0.43
FAP Q12884 1/20 0.43
DPP8 Q6V1X1 1/20 0.43
DPP9 Q86TI2 1/20 0.43
CHRM3 P20309 1/20 0.42
ALDH1A1 P00352 1/20 0.42
HSD11B1 P28845 1/20 0.41
DRD4 P21917 1/20 0.41
OPRM1 P35372 1/20 0.41
OPRL1 P41146 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL2329416 0.99 SIRT2 (0.45) SIRT2SIRT1EPHX1ROCK2ROCK1
Hydrochloric Acid SCHEMBL2329419 0.99 SIRT2 (0.45) SIRT2SIRT1EPHX1ROCK2ROCK1
SCHEMBL7415900 0.96 SIRT2 (0.47) SIRT2SIRT1EPHX1ROCK2ROCK1
SCHEMBL7419120 0.91 SIRT2 (0.48) SIRT2SIRT1EPHX1ROCK2ROCK1
SCHEMBL7482530 0.91 SIRT2 (0.48) SIRT2SIRT1EPHX1ROCK2ROCK1
Hydrochloric Acid SCHEMBL2327307 0.90 SIRT2 (0.47) SIRT2SIRT1ROCK2ROCK1DPP4
Hydrochloric Acid SCHEMBL7424649 0.90 SIRT2 (0.47) SIRT2SIRT1ROCK2ROCK1DPP4
Hydrochloric Acid SCHEMBL2327302 0.90 SIRT2 (0.47) SIRT2SIRT1ROCK2ROCK1DPP4
Trifluoroacetic Acid SCHEMBL2330275 0.87 GPR6 (0.47) SIRT2SIRT1EPHX1ROCK2ROCK1
Methylene Chloride SCHEMBL27479070 0.87 SIRT2 (0.45) SIRT2SIRT1ROCK2ROCK1DPP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0853618-A4 SUBSTITUTED (SULFINIC ACID, SULFONIC ACID, SULFONYLAMINO OR SULFINYLAMINO) N- (AMINOIMINOMETHYL)PHENYLALKYL]-AZAHETEROCYCLYLAMIDE COMPOUNDS RHONE POULENC RORER PHARMA (US) 2000-03-15 EP disclosed
EP-0853618-A1 SUBSTITUTED (SULFINIC ACID, SULFONIC ACID, SULFONYLAMINO OR SULFINYLAMINO) N- (AMINOIMINOMETHYL)PHENYLALKYL]-AZAHETEROCYCLYLAMIDE COMPOUNDS RHONE-POULENC RORER PHARMACEUTICALS, INC. (US) 1998-07-22 EP disclosed
US-5612353-A ANTICOAGULANT RHONE-POULENC RORER PHARMACEUTICALS INC. (US) 1997-03-18 US disclosed
WO-1996040679-A1 SUBSTITUTED (SULFINIC ACID, SULFONIC ACID, SULFONYLAMINO OR SULFINYLAMINO) N-[(AMINOIMINOMETHYL)PHENYLALKYL]-AZAHETEROCYCLYLAMIDE COMPOUNDS RHÔNE-POULENC RORER PHARMACEUTICALS INC. (US) 1996-12-19 WO disclosed