SCHEMBL7420330

SCHEMBL7420330

Brc1nccs1.C(#CC1CCCCC1)c1nccs1

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 4/20 0.42
CYP1A2 P05177 1/20 0.42
MEN1 O00255 1/20 0.35
TSHR P16473 1/20 0.35
KMT2A Q03164 1/20 0.35
KCNH2 Q12809 1/20 0.33
POLB P06746 2/20 0.33
HTT P42858 1/20 0.32
EPHX2 P34913 1/20 0.32
KDM4E B2RXH2 1/20 0.32
PDGFRB P09619 1/20 0.32
PDGFRA P16234 1/20 0.32
RBBP9 O75884 1/20 0.32
IDO1 P14902 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7419628 0.92 GRM5 (0.41) GRM5CYP1A2MEN1KMT2AHTT
SCHEMBL4861899 0.92 GRM5 (0.47) GRM5CYP1A2MEN1TSHRKMT2A
SCHEMBL7385448 0.84 GRM5 (0.47) GRM5CYP1A2MEN1TSHRKMT2A
SCHEMBL7388499 0.71 GRM5 (0.39) GRM5MEN1TSHRKMT2AHTT
SCHEMBL4861917 0.69 POLB (0.43) GRM5MEN1TSHRKMT2APOLB
SCHEMBL15870993 0.68 GRM5 (0.68) GRM5TSHR
SCHEMBL6063 0.67
SCHEMBL30278460 0.66 PDPK1 (0.45) GRM5CYP1A2
Bromide SCHEMBL5403925 0.65
SCHEMBL7608425 0.65

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1214303-A1 HETEROCYCLIC COMPOUNDS AND METHODS OF USE THEREOF Merck & Co., Inc. (US) 2002-06-19 EP disclosed
WO-2001016121-A1 HETEROCYCLIC COMPOUNDS AND METHODS OF USE THEREOF MERCK & CO., INC. (US) 2001-03-08 WO disclosed