Chloramben

Chloramben

SCHEMBL7422202

Nc1cc(Cl)cc(C(=O)O)c1Cl.[NaH]

nearest known ligand 0.96

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.96
AKR1C4 P17516 1/20 0.48
AKR1C3 P42330 1/20 0.48
AKR1C2 P52895 1/20 0.48
AKR1C1 Q04828 1/20 0.48
ALDH1A1 P00352 4/20 0.45
TP53 P04637 1/20 0.45
HPGD P15428 2/20 0.44
HSD17B10 Q99714 1/20 0.44
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
TPMT P51580 1/20 0.41
DYRK1A Q13627 1/20 0.41
KMT2A Q03164 4/20 0.41
KDM4E B2RXH2 4/20 0.41
TSHR P16473 1/20 0.41
CASP1 P29466 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
GFER P55789 1/20 0.41
RXFP1 Q9HBX9 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Chloramben SCHEMBL117283 0.98 CYP3A4 (1.00) CYP3A4AKR1C4AKR1C3AKR1C2AKR1C1
Chloramben SCHEMBL55091 0.98 CYP3A4 (1.00) CYP3A4AKR1C4AKR1C3AKR1C2AKR1C1
Chloramben SCHEMBL29448826 0.98 CYP3A4 (1.00) CYP3A4AKR1C4AKR1C3AKR1C2AKR1C1
Chloramben SCHEMBL164009 0.96 CYP3A4 (0.96) CYP3A4AKR1C4AKR1C3AKR1C2AKR1C1
Chloramben SCHEMBL11298879 0.96 CYP3A4 (0.96) CYP3A4AKR1C4AKR1C3AKR1C2AKR1C1
Chloramben SCHEMBL11629597 0.96 CYP3A4 (0.96) CYP3A4AKR1C4AKR1C3AKR1C2AKR1C1
Chloramben SCHEMBL163142 0.94 CYP3A4 (0.92) CYP3A4AKR1C4AKR1C3AKR1C2AKR1C1
Chloramben SCHEMBL11010427 0.90 CYP3A4 (0.85) CYP3A4AKR1C4AKR1C3AKR1C2AKR1C1
3,5-Dichloroanthranilic Acid SCHEMBL6036778 0.87 CYP3A4 (0.79) CYP3A4AKR1C4AKR1C3AKR1C2AKR1C1
Chloramben SCHEMBL22042184 0.83 CYP3A4 (0.72) CYP3A4AKR1C4AKR1C3AKR1C2AKR1C1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023099381-A1 (1,4,5-TRISUBSTITUTED-1H-PYRAZOLE-3-YL)OXY-2-ALKOXYTHIO ALKYL ACIDS AND DERIVATIVES THEREOF, THEIR SALTS AND THEIR USE AS HERBICIDAL ACTIVE AGENTS BAYER AKTIENGESELLSCHAFT (DE) 2023-06-08 WO disclosed
EP-0719244-A1 PROCESS OF PREPARING 2,3,5-TRIHALOBENZALDEHYDE THE WELLCOME FOUNDATION LIMITED (GB) 1996-07-03 EP disclosed
WO-1995007877-A1 PROCESS OF PREPARING 2,3,5-TRIHALOBENZALDEHYDE THE WELLCOME FOUNDATION LIMITED (GB) 1995-03-23 WO disclosed