SCHEMBL7423476

SCHEMBL7423476

Cn1c(CNc2ccc(C#N)cc2)nc2cc(C(CCCl)C(=O)C3CCCC3)ccc21

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITK Q08881 3/20 0.47
HDAC6 Q9UBN7 4/20 0.41
NPC1 O15118 4/20 0.41
KDM4E B2RXH2 2/20 0.41
AURKA O14965 1/20 0.41
MAP4K4 O95819 1/20 0.41
CHEK2 O96017 1/20 0.41
PRKCG P05129 1/20 0.41
PHKG2 P15735 1/20 0.41
MARK3 P27448 1/20 0.41
FLT3 P36888 1/20 0.41
CSNK1A1 P48729 1/20 0.41
CSNK1D P48730 1/20 0.41
CLK2 P49760 1/20 0.41
GSK3B P49841 1/20 0.41
IRAK1 P51617 1/20 0.41
RPS6KA3 P51812 1/20 0.41
NEK4 P51957 1/20 0.41
CSNK1G2 P78368 1/20 0.41
MAP4K2 Q12851 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7410722 0.86 F2 (0.53) HDAC6F2F10PRSS1PRSS2
SCHEMBL7423473 0.83 ITK (0.47) ITKAURKAMAP4K4CHEK2PRKCG
SCHEMBL4937046 0.79 F2 (0.49) ITKHDAC6NPC1KDM4EALDH1A1
SCHEMBL4937057 0.79 F2 (0.49) ITKHDAC6NPC1KDM4EALDH1A1
SCHEMBL7412219 0.77 F2 (0.55) ITKHDAC6NPC1KDM4EAURKA
SCHEMBL7418283 0.76 F2 (0.49) ITKHDAC6NPC1KDM4EALDH1A1
SCHEMBL14914339 0.74 HDAC6 (0.51) HDAC6NPC1KDM4EALDH1A1RAB9A
SCHEMBL7415541 0.74 F2 (0.48) ITKHDAC6NPC1KDM4EF2
SCHEMBL30937423 0.73 HDAC6 (0.62) HDAC6NPC1KDM4EF2F10
SCHEMBL28088312 0.73 HDAC6 (0.62) HDAC6NPC1KDM4EF2F10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1095025-B1 BENZIMIDAZOLES, PRODUCTION THEREOF AND USE THEREOF AS MEDICAMENTS BOEHRINGER INGELHEIM PHARMA (DE) 2002-12-11 EP disclosed
US-6248770-B1 CARDIOVASCULAR DISORDERS BOEHRINGER INGELHEIM PHARMA KG (DE) 2001-06-19 US disclosed