SCHEMBL742487

SCHEMBL742487

COCCCn1c([C@@H]2CCCN(C(=O)C[C@@H](Cc3ccc4ccccc4c3)N(C(=O)O)C(C)(C)C)C2)nc2cccc(C)c21

nearest known ligand 0.36

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 5/20 0.36
KCNH2 Q12809 5/20 0.36
CYP2D6 P10635 4/20 0.36
PPARA Q07869 1/20 0.34
ALDH1A1 P00352 4/20 0.34
TSHR P16473 3/20 0.34
CHRM1 P11229 1/20 0.33
LMNA P02545 1/20 0.33
HTT P42858 1/20 0.33
KMT2A Q03164 1/20 0.32
PROKR1 Q8TCW9 2/20 0.32
TACR1 P25103 1/20 0.32
BTK Q06187 2/20 0.32
CYP3A4 P08684 1/20 0.32
LSS P48449 1/20 0.32
BCHE P06276 1/20 0.31
OPRD1 P41143 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL741454 0.93 HRH1 (0.36) HRH1KCNH2CYP2D6PPARAALDH1A1
SCHEMBL741317 0.91 HRH1 (0.45) HRH1KCNH2CYP2D6CHRM1PROKR1
SCHEMBL741747 0.90 HRH1 (0.36) HRH1KCNH2CYP2D6PPARAALDH1A1
SCHEMBL738741 0.87 KCNH2 (0.39) HRH1KCNH2CYP2D6ALDH1A1TSHR
SCHEMBL742065 0.87 HRH1 (0.39) HRH1KCNH2CYP2D6PPARACHRM1
SCHEMBL742192 0.87 HRH1 (0.40) HRH1KCNH2CYP2D6CHRM1
SCHEMBL740611 0.87 KCNH2 (0.38) HRH1KCNH2CYP2D6PPARACHRM1
SCHEMBL740700 0.87 KCNH2 (0.36) HRH1KCNH2CYP2D6ALDH1A1TSHR
SCHEMBL740699 0.87 KCNH2 (0.36) HRH1KCNH2CYP2D6ALDH1A1TSHR
SCHEMBL742676 0.86 CYP2D6 (0.34) HRH1KCNH2CYP2D6PPARAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed