SCHEMBL7426499

SCHEMBL7426499

COc1cc(C#N)nc(C#N)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NQO1 P15559 1/20 0.53
KDM4E B2RXH2 6/20 0.51
MAPT P10636 3/20 0.47
GAA P10253 3/20 0.47
ALDH1A1 P00352 6/20 0.46
HPGD P15428 4/20 0.45
TSHR P16473 2/20 0.45
MAPK1 P28482 2/20 0.45
L3MBTL1 Q9Y468 2/20 0.45
HSD17B10 Q99714 2/20 0.45
LMNA P02545 1/20 0.45
CASP1 P29466 1/20 0.45
CASP7 P55210 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
HPGDS O60760 1/20 0.44
POLB P06746 2/20 0.42
PTBP1 P26599 1/20 0.42
ADORA1 P30542 1/20 0.42
USP8 P40818 2/20 0.41
PPARG P37231 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7227326 0.87 TSHR (0.49) NQO1KDM4EMAPTGAAALDH1A1
SCHEMBL2088644 0.86 NQO1 (0.46) NQO1KDM4EMAPTGAAALDH1A1
SCHEMBL26986651 0.86 NQO1 (0.46) NQO1KDM4EMAPTGAAALDH1A1
SCHEMBL7048544 0.86 KDM4E (0.53) NQO1KDM4EMAPTGAAALDH1A1
SCHEMBL20412651 0.77 CCR1 (0.62) NQO1KDM4EMAPTGAAALDH1A1
SCHEMBL21121957 0.76 PDE2A (0.59) NQO1KDM4EALDH1A1LMNAPOLB
SCHEMBL5225009 0.76 GAA (0.42) NQO1KDM4EMAPTGAAALDH1A1
Caerulomycinonitrile SCHEMBL8515198 0.75 HSP90AA1 (0.54) KDM4EMAPTGAAALDH1A1L3MBTL1
SCHEMBL503826 0.74 CCR1 (0.55) NQO1KDM4EMAPTALDH1A1MAPK1
SCHEMBL29705335 0.74 NQO1 (0.43) NQO1KDM4EMAPTGAAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002068417-A3 HETEROPOLYCYCLIC COMPOUNDS AND THEIR USE AS METABOTROPIC GLUTAMATE RECEPTOR ANTAGONISTS SLASSI ABDELMALIK (CA) 2002-11-14 WO disclosed