SCHEMBL7429070

SCHEMBL7429070

CC(C)(C)OC(=O)NCCCOCc1ccccc1N

nearest known ligand 0.49

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CA1 P00915 9/20 0.49
CA2 P00918 9/20 0.49
CA12 O43570 6/20 0.49
CA9 Q16790 6/20 0.49
NQO2 P16083 1/20 0.45
IDO1 P14902 1/20 0.44
TDP1 Q9NUW8 1/20 0.43
MAOA P21397 1/20 0.42
MAOB P27338 1/20 0.42
DRD2 P14416 3/20 0.42
MEN1 O00255 1/20 0.42
GAA P10253 1/20 0.42
KMT2A Q03164 1/20 0.42
MALT1 Q9UDY8 1/20 0.41
HDAC1 Q13547 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15584098 0.92 IDO1 (0.48) CA1CA2CA12CA9NQO2
SCHEMBL10705964 0.84 CA1 (0.46) CA1CA2CA12CA9NQO2
SCHEMBL7531330 0.84 NQO2 (0.48) CA1CA2CA12CA9NQO2
SCHEMBL27770724 0.83 TDP1 (0.50) CA1CA2CA12CA9NQO2
SCHEMBL13622021 0.82 IDO1 (0.56) CA1CA2CA12CA9IDO1
SCHEMBL31250995 0.81 NQO2 (0.56) CA1CA2CA12CA9NQO2
SCHEMBL1231492 0.81 NQO2 (0.56) CA1CA2CA12CA9NQO2
SCHEMBL2061998 0.78 KCNA5 (0.54) CA1CA12NQO2IDO1MALT1
SCHEMBL22163551 0.78 CA12 (0.40) CA1CA2CA12CA9NQO2
SCHEMBL29450820 0.78 CA12 (0.40) CA1CA2CA12CA9NQO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1208104-A2 TRICYCLIC INHIBITORS OF POLY(ADP-RIBOSE) POLYMERASES AGOURON PHARMACEUTICALS, INC. (US) 2002-05-29 EP disclosed
WO-2001016136-A2 TRICYCLIC INHIBITORS OF POLY(ADP-RIBOSE) POLYMERASES AGOURON PHARMACEUTICALS, INC. (US) 2001-03-08 WO disclosed