SCHEMBL7429172

SCHEMBL7429172

NCc1ccc(C(=O)Oc2ccc(C(=O)O)cc2)cc1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRSS1 P07477 4/20 0.66
F2 P00734 2/20 0.66
PRSS2 P07478 2/20 0.66
PRSS3 P35030 2/20 0.66
LOXL2 Q9Y4K0 2/20 0.56
PARP10 Q53GL7 1/20 0.53
KLK1 P06870 2/20 0.51
TMPRSS2 O15393 1/20 0.51
RXRA P19793 3/20 0.49
RXRB P28702 3/20 0.49
ALDH1A1 P00352 1/20 0.48
SRD5A2 P31213 1/20 0.47
HSD17B10 Q99714 2/20 0.46
NR4A2 P43354 3/20 0.45
NPC1 O15118 1/20 0.45
POLB P06746 1/20 0.45
RAB9A P51151 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
NR4A1 P22736 1/20 0.45
NR4A3 Q92570 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Propane SCHEMBL27557200 0.95 PRSS1 (0.61) PRSS1F2PRSS2PRSS3LOXL2
Propane SCHEMBL8503848 0.95 PRSS1 (0.61) PRSS1F2PRSS2PRSS3LOXL2
SCHEMBL27650063 0.88 PRSS1 (0.63) PRSS1F2PRSS2PRSS3LOXL2
SCHEMBL16180747 0.88 PARP10 (0.64) PRSS1F2PRSS2PRSS3LOXL2
SCHEMBL22688039 0.86 PRSS1 (0.66) PRSS1F2PRSS2PRSS3LOXL2
Hydrochloric Acid SCHEMBL7426558 0.86 PRSS1 (0.61) PRSS1F2PRSS2PRSS3LOXL2
SCHEMBL4597931 0.85 PARP10 (0.62) PRSS1F2PRSS2PRSS3PARP10
SCHEMBL7536846 0.85 PARP10 (0.62) PRSS1F2PRSS2PRSS3PARP10
SCHEMBL376498 0.85 PARP10 (0.62) PRSS1F2PRSS2PRSS3PARP10
SCHEMBL16180672 0.85 PRSS1 (0.64) PRSS1F2PRSS2PRSS3LOXL2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1073624-A1 AMINOMETHYL-BENZOIC ESTER DERIVATIVES AS TRYPTASE INHIBITORS Proteus Molecular Design Limited (GB) 2001-02-07 EP disclosed
WO-1999055661-A1 AMINOMETHYL-BENZOIC ESTER DERIVATIVES AS TRYPTASE INHIBITORS PROTEUS MOLECULAR DESIGN LIMITED (GB) 1999-11-04 WO disclosed