SCHEMBL7429689

SCHEMBL7429689

CCCOC(=O)C1=C(C)NC(CF)=C(C(=O)OC)C1c1cccc(Cl)c1Cl

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 3/20 0.72
ABCB11 O95342 3/20 0.72
CYP3A4 P08684 3/20 0.72
TBXA2R P21731 3/20 0.72
ADRA1A P35348 3/20 0.72
SLC6A3 Q01959 3/20 0.72
KDM4E B2RXH2 2/20 0.72
MEN1 O00255 2/20 0.72
CYP1A2 P05177 2/20 0.72
CYP2C19 P33261 2/20 0.72
KMT2A Q03164 2/20 0.72
HIF1A Q16665 2/20 0.72
HSD17B10 Q99714 2/20 0.72
ABCB1 P08183 2/20 0.72
ADORA3 P0DMS8 2/20 0.72
ADRB3 P13945 2/20 0.72
OPRK1 P41145 2/20 0.72
SCN5A Q14524 2/20 0.72
NR1I2 O75469 2/20 0.72
TSHR P16473 2/20 0.72

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7438922 0.94 CYP2C9 (0.62) CYP2C9ABCB11CYP3A4TBXA2RADRA1A
SCHEMBL7429576 0.93 CYP2C9 (0.68) CYP2C9ABCB11CYP3A4TBXA2RADRA1A
SCHEMBL7318977 0.89 CYP2C9 (0.68) CYP2C9ABCB11CYP3A4TBXA2RADRA1A
SCHEMBL7428072 0.89 CYP2C9 (0.56) CYP2C9ABCB11CYP3A4TBXA2RADRA1A
SCHEMBL7434261 0.87 CYP2C9 (0.55) CYP2C9ABCB11CYP3A4TBXA2RADRA1A
SCHEMBL7434919 0.86 CYP2C9 (0.65) CYP2C9ABCB11CYP3A4TBXA2RADRA1A
SCHEMBL7439079 0.86 CYP2C9 (0.69) CYP2C9ABCB11CYP3A4TBXA2RADRA1A
SCHEMBL7431523 0.85 TBXA2R (0.54) CYP2C9ABCB11CYP3A4TBXA2RADRA1A
SCHEMBL9501593 0.85 KDM4E (0.85) CYP2C9ABCB11CYP3A4TBXA2RADRA1A
SCHEMBL7429568 0.85 CYP2C9 (0.64) CYP2C9ABCB11CYP3A4TBXA2RADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0125803-A2 Pharmaceutically active dihydropyridines FISONS plc (GB) 1984-11-21 EP claimed
EP-0125803-A2 Pharmaceutically active dihydropyridines FISONS plc (GB) 1984-11-21 EP disclosed