SCHEMBL7433357

SCHEMBL7433357

CCOC(=O)C(CCc1ccccc1)NC1CSc2ccccc2N(CC(=O)O)C1=O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ACE P12821 8/20 0.81
ABCB11 O95342 1/20 0.70
AGTR2 P50052 1/20 0.70
PDE3A Q14432 1/20 0.70
TDP1 Q9NUW8 1/20 0.70
KDM4E B2RXH2 1/20 0.69
CYP3A4 P08684 1/20 0.69
MME P08473 2/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10853559 1.00 ACE (0.81) ACEABCB11AGTR2PDE3ATDP1
SCHEMBL10855240 1.00 ACE (0.81) ACEABCB11AGTR2PDE3ATDP1
SCHEMBL10853549 1.00 ACE (0.81) ACEABCB11AGTR2PDE3ATDP1
Hydrochloric Acid SCHEMBL11013211 0.99 ACE (0.80) ACEABCB11AGTR2PDE3ATDP1
Hydrochloric Acid SCHEMBL9824878 0.99 ACE (0.80) ACEABCB11AGTR2PDE3ATDP1
Hydrochloric Acid SCHEMBL10856588 0.99 ACE (0.80) ACEABCB11AGTR2PDE3ATDP1
Hydrochloric Acid SCHEMBL9824873 0.99 ACE (0.80) ACEABCB11AGTR2PDE3ATDP1
SCHEMBL10856359 0.96 ACE (0.74) ACEABCB11AGTR2PDE3ATDP1
SCHEMBL10856344 0.96 ACE (0.74) ACEABCB11AGTR2PDE3ATDP1
SCHEMBL11012582 0.94 ACE (0.71) ACEABCB11AGTR2PDE3ATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4539150-A HYPOTENSIVE AGENTS, SULFIDING, CYCLIZATION MITSUI TOATSU CHEMICALS, INC. (JP) 1985-09-03 US claimed
US-4477464-A Hetero-benzazepine derivatives and their pharmaceutical use CIBA-GEIGY CORPORATION (US) 1984-10-16 US claimed
US-4539150-A HYPOTENSIVE AGENTS, SULFIDING, CYCLIZATION MITSUI TOATSU CHEMICALS, INC. (JP) 1985-09-03 US disclosed
EP-0120728-A1 Thiazine and thiazepine containing compounds E.R. Squibb & Sons, Inc. (US) 1984-10-03 EP disclosed