SCHEMBL7433914

SCHEMBL7433914

CN1CCN(C(=O)c2ccc(-c3nnn(CC(=O)C(CC(=O)OC(C)(C)C)NC(=O)OCc4ccccc4)n3)cc2)CC1

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47
ALDH1A1 P00352 2/20 0.43
MAPT P10636 1/20 0.43
ESR2 Q92731 1/20 0.43
AVPR2 P30518 2/20 0.42
AVPR1A P37288 2/20 0.42
TGM2 P21980 2/20 0.41
TP53 P04637 2/20 0.41
POLB P06746 1/20 0.41
P2RX7 Q99572 5/20 0.40
CYP3A4 P08684 1/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
P2RY12 Q9H244 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7433569 0.91 CYP1A2 (0.49) CYP1A2CYP2C9CYP2C19AVPR2AVPR1A
Hydrochloric Acid SCHEMBL7429640 0.90 CYP1A2 (0.48) CYP1A2CYP2C9CYP2C19AVPR2AVPR1A
SCHEMBL7437630 0.90 CYP1A2 (0.56) CYP1A2CYP2C9CYP2C19ALDH1A1MAPT
SCHEMBL7438698 0.90 CYP1A2 (0.58) CYP1A2CYP2C9CYP2C19ALDH1A1MAPT
SCHEMBL7437704 0.89 CYP1A2 (0.53) CYP1A2CYP2C9CYP2C19ALDH1A1MAPT
SCHEMBL7440422 0.88 CYP1A2 (0.52) CYP1A2CYP2C9CYP2C19ALDH1A1MAPT
SCHEMBL7439105 0.87 CYP1A2 (0.51) CYP1A2CYP2C9CYP2C19ALDH1A1MAPT
SCHEMBL7431018 0.84 CYP1A2 (0.51) CYP1A2CYP2C9CYP2C19ALDH1A1TP53
SCHEMBL7483493 0.84 CYP1A2 (0.52) CYP1A2CYP2C9CYP2C19TP53MEN1
SCHEMBL7431049 0.83 CYP1A2 (0.49) CYP1A2CYP2C9CYP2C19ALDH1A1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5710153-A INTERLEUKIN CONVERTING ENZYME INHIBITORS ONO PHRAMACEUTICAL CO., LTD. (JP) 1998-01-20 US disclosed
EP-0761680-A2 Tetrazole compounds having Interleukin-1beta converting enzyme inhibitory activity ONO PHARMACEUTICAL CO., LTD. (JP) 1997-03-12 EP disclosed