SCHEMBL7439697

SCHEMBL7439697

O=C(O)C(Cc1ccccc1)CC(Cc1ccccc1)C(=O)O

nearest known ligand 0.86

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.86
SLC1A3 P43003 1/20 0.78
SLC1A2 P43004 1/20 0.78
SLC1A1 P43005 1/20 0.78
CPA1 P15085 7/20 0.73
CPA3 P15088 3/20 0.73
FOLH1 Q04609 3/20 0.73
CPB1 P15086 1/20 0.73
CPB2 Q96IY4 1/20 0.73
NAALAD2 Q9Y3Q0 1/20 0.70

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7432418 1.00 CYP1A2 (0.86) CYP1A2SLC1A3SLC1A2SLC1A1CPA1
SCHEMBL9622038 1.00 CYP1A2 (0.86) CYP1A2SLC1A3SLC1A2SLC1A1CPA1
SCHEMBL4664822 0.93 CYP1A2 (1.00) CYP1A2SLC1A3SLC1A2SLC1A1CPA1
SCHEMBL9875948 0.91 CYP1A2 (0.95) CYP1A2SLC1A3SLC1A2SLC1A1CPA1
SCHEMBL22115491 0.91 CYP1A2 (0.95) CYP1A2SLC1A3SLC1A2SLC1A1CPA1
SCHEMBL27291058 0.91 CYP1A2 (0.95) CYP1A2SLC1A3SLC1A2SLC1A1CPA1
SCHEMBL3928753 0.90 CYP1A2 (0.70) CYP1A2SLC1A3SLC1A2SLC1A1CPA1
SCHEMBL4021013 0.90 CYP1A2 (0.70) CYP1A2SLC1A3SLC1A2SLC1A1CPA1
SCHEMBL19821208 0.88 CYP1A2 (0.83) CYP1A2SLC1A3SLC1A2SLC1A1CPA1
SCHEMBL6724759 0.88 CYP1A2 (0.83) CYP1A2SLC1A3SLC1A2SLC1A1CPA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5166212-A Hypotensive agents, analgesics CIBA-GEIGY CORPORATION (US) 1992-11-24 US disclosed
US-5096925-A N-substituted butyramide derivatives CIBA-GEIGY CORPORATION (US) 1992-03-17 US disclosed
US-5021430-A Enkephalinase inhibitors, analgesics, hypotensives CIBA-GEIGY CORPORATION (US) 1991-06-04 US disclosed
US-4939261-A ANALGESICS, ANTIDEPRESSANTS, HYPOTENSIVE AGENTS, NEUROLEPTIC AGENTS CIBA-GEIGY CORPORATION (US) 1990-07-03 US disclosed
EP-0185079-B1 N-SUBSTITUTED BUTYRAMIDE DERIVATIVES CIBA-GEIGY AG (CH) 1988-10-19 EP disclosed
EP-0225292-A2 Certain N-substituted butyramide derivatives CIBA-GEIGY AG (CH) 1987-06-10 EP disclosed
EP-0185079-A1 CIBA GEIGY AG 1986-06-25 EP disclosed
WO-1986000066-A1 N-SUBSTITUTED BUTYRAMIDE DERIVATIVES CIBA-GEIGY AG (CH) 1986-01-03 WO disclosed