SCHEMBL7440449

SCHEMBL7440449

O=C(O)CC(NC(=O)OCc1ccccc1)C(=O)Cn1nnc(-c2cccc(-c3ccccc3)c2)n1

nearest known ligand 0.54

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.54
CYP2C9 P11712 1/20 0.54
CYP2C19 P33261 1/20 0.54
ALDH1A1 P00352 1/20 0.52
LMNA P02545 1/20 0.52
HTT P42858 1/20 0.52
SMN1; SMN2 Q16637 1/20 0.52
TDP1 Q9NUW8 1/20 0.52
CASP1 P29466 17/20 0.51
TP53 P04637 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7429152 0.93 CYP1A2 (0.60) CYP1A2CYP2C9CYP2C19CASP1TP53
SCHEMBL7435530 0.93 CYP1A2 (0.63) CYP1A2CYP2C9CYP2C19CASP1TP53
SCHEMBL7432223 0.93 SMN1; SMN2 (0.55) CYP1A2CYP2C9CYP2C19ALDH1A1LMNA
SCHEMBL7434939 0.90 SMN1; SMN2 (0.57) CYP1A2CYP2C9CYP2C19ALDH1A1LMNA
SCHEMBL7427222 0.89 SMN1; SMN2 (0.52) CYP1A2CYP2C9CYP2C19ALDH1A1LMNA
SCHEMBL7431018 0.89 CYP1A2 (0.51) CYP1A2CYP2C9CYP2C19ALDH1A1LMNA
SCHEMBL7685015 0.89 CYP1A2 (0.57) CYP1A2CYP2C9CYP2C19HTTCASP1
SCHEMBL7432412 0.89 CYP1A2 (0.57) CYP1A2CYP2C9CYP2C19CASP1TP53
Hydrochloric Acid SCHEMBL7696612 0.88 CYP1A2 (0.56) CYP1A2CYP2C9CYP2C19HTTCASP1
SCHEMBL7426313 0.87 CYP1A2 (0.53) CYP1A2CYP2C9CYP2C19CASP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5710153-A INTERLEUKIN CONVERTING ENZYME INHIBITORS ONO PHRAMACEUTICAL CO., LTD. (JP) 1998-01-20 US claimed
EP-0761680-A2 Tetrazole compounds having Interleukin-1beta converting enzyme inhibitory activity ONO PHARMACEUTICAL CO., LTD. (JP) 1997-03-12 EP claimed
US-5710153-A INTERLEUKIN CONVERTING ENZYME INHIBITORS ONO PHRAMACEUTICAL CO., LTD. (JP) 1998-01-20 US disclosed
EP-0761680-A2 Tetrazole compounds having Interleukin-1beta converting enzyme inhibitory activity ONO PHARMACEUTICAL CO., LTD. (JP) 1997-03-12 EP disclosed