SCHEMBL7443170

SCHEMBL7443170

CCOC(=O)NCC(=O)c1ccc(O)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 2/20 0.56
CA12 O43570 2/20 0.56
CA1 P00915 2/20 0.56
CA2 P00918 2/20 0.56
CA7 P43166 2/20 0.56
CA9 Q16790 2/20 0.56
CA14 Q9ULX7 2/20 0.56
ESR2 Q92731 1/20 0.56
HSD17B3 P37058 8/20 0.49
MIF P14174 1/20 0.48
ALDH1A1 P00352 2/20 0.47
NPC1 O15118 2/20 0.47
RAB9A P51151 2/20 0.47
MAPT P10636 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.46
CHRM1 P11229 1/20 0.45
TSHR P16473 1/20 0.45
SLC6A2 P23975 1/20 0.45
KDR P35968 1/20 0.45
TDP1 Q9NUW8 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Methane SCHEMBL9836231 0.98 ESR1 (0.54) ESR1CA12CA1CA2CA7
SCHEMBL10740037 0.85 SMN1; SMN2 (0.60) CA12CA1CA2CA9ALDH1A1
SCHEMBL10782158 0.85 KMT2A (0.54) ALDH1A1NPC1RAB9AMAPTSMN1; SMN2
SCHEMBL20524444 0.84 KMT2A (0.60) CA12CA1CA2CA9ALDH1A1
Methane SCHEMBL11375164 0.83 KMT2A (0.53) ALDH1A1NPC1RAB9AMAPTSMN1; SMN2
SCHEMBL10805330 0.81 HDAC3 (0.58) ALDH1A1RAB9AMAPTSMN1; SMN2TDP1
SCHEMBL10459828 0.81 CA12 (0.46) ESR1CA12CA1CA2CA7
SCHEMBL10457925 0.79 SMN1; SMN2 (0.48) ESR1CA12CA1CA2CA7
SCHEMBL2009324 0.79 NR1H4 (0.47) CA12CA1CA2CA7CA9
SCHEMBL9837130 0.78 PTPN1 (0.52) ESR1CA12CA1CA2CA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0238357-B1 1,2,4-TRIAZINONE DERIVATIVES, THEIR PREPARATION AND USE Sankyo Company Limited (JP) 1991-05-29 EP disclosed
US-4898862-A 1,2,4-triazinone derivatives, their preparation and use SANKYO COMPANY LIMITED (JP) 1990-02-06 US disclosed
EP-0238357-A2 1,2,4-Triazinone derivatives, their preparation and use Sankyo Company Limited (JP) 1987-09-23 EP disclosed
US-4453003-A ENZYME INHIBITORS, ANTIINFLAMMATORY AGENTS UMEZAWA HAMAO (JP) 1984-06-05 US disclosed
US-4391986-A Process for producing threo-3-amino-2-hydroxybutanoyl-aminoacetic acids, as well as novel intermediates therefor and process for producing them NIPPON KAYAKU KABUSHIKI KAISHA (JP) 1983-07-05 US disclosed
US-4281180-A Process for producing threo-3-amino-2-hydroxybutanoyl-aminoacetic acids, as well as novel intermediated therefor and process for producing them NIPPON KAYAKU KABUSHIKI KAISHA (JP) 1981-07-28 US disclosed