SCHEMBL744375

SCHEMBL744375

CN1C2CCC1C(c1cncc(-c3ccc4[nH]c(C(F)(F)F)cc4c3)c1)C(N/C(=C/C(=O)O)C(=O)O)C2

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 4/20 0.40
KCNH2 Q12809 4/20 0.40
CHRNB2 P17787 2/20 0.34
CHRNA4 P43681 1/20 0.34
DYRK1A Q13627 6/20 0.34
WNT1 P04628 2/20 0.34
GSK3B P49841 1/20 0.31
CHRNA6 Q15825 1/20 0.31
SLC6A2 P23975 1/20 0.31
SLC6A4 P31645 1/20 0.31
SLC6A3 Q01959 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Fumaric Acid SCHEMBL989196 0.73 CHRNA7 (0.43) CHRNA7KCNH2CHRNB2CHRNA4DYRK1A
Fumaric Acid SCHEMBL989195 0.73 CHRNA7 (0.43) CHRNA7KCNH2CHRNB2CHRNA4DYRK1A
SCHEMBL748444 0.70 CHRNA7 (0.48) CHRNA7KCNH2CHRNB2CHRNA4DYRK1A
SCHEMBL744853 0.70 CHRNA7 (0.48) CHRNA7KCNH2CHRNB2CHRNA4DYRK1A
Fumaric Acid SCHEMBL747023 0.64 CHRNA7 (0.47) CHRNA7KCNH2SLC6A2SLC6A3
Trifluoroacetic Acid SCHEMBL744720 0.63 CHRNA7 (0.47) CHRNA7KCNH2CHRNB2CHRNA4DYRK1A
Trifluoroacetic Acid SCHEMBL4114805 0.63 KCNH2 (0.45) CHRNA7KCNH2CHRNB2CHRNA4DYRK1A
SCHEMBL744858 0.62 KCNH2 (0.56) CHRNA7KCNH2CHRNB2CHRNA4SLC6A2
SCHEMBL989197 0.62 CHRNA7 (0.39) CHRNA7KCNH2DYRK1AWNT1GSK3B
Trifluoroacetic Acid SCHEMBL747090 0.61 CHRNA7 (0.51) CHRNA7KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2431368-A1 CNS active fused bicycloheterocycle substituted azabicyclic alkane derivatives Abbott Laboratories (US) 2012-03-21 EP disclosed