SCHEMBL7444973

SCHEMBL7444973

NCCCC1Cc2ccccc2C1

nearest known ligand 0.58

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 5/20 0.58
HRH1 P35367 3/20 0.58
IDO1 P14902 3/20 0.55
CYP19A1 P11511 1/20 0.41
RET P07949 1/20 0.41
HTR2C P28335 1/20 0.41
CYP2D6 P10635 2/20 0.38
SLC6A2 P23975 2/20 0.38
SLC6A4 P31645 2/20 0.38
CYP2C19 P33261 2/20 0.38
SLC6A3 Q01959 2/20 0.38
KCNH2 Q12809 2/20 0.38
GBA1 P04062 1/20 0.38
PLAU P00749 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8300848 0.92 IDO1 (0.56) HTR2AHRH1IDO1CYP19A1RET
SCHEMBL31536940 0.86 IDO1 (0.59) HTR2AHRH1IDO1CYP19A1RET
SCHEMBL6992991 0.86 IDO1 (0.59) HTR2AHRH1IDO1CYP19A1RET
Hydrochloric Acid SCHEMBL7212472 0.84 IDO1 (0.62) HTR2AHRH1IDO1CYP19A1RET
SCHEMBL10530881 0.78 IDO1 (0.50) HTR2AHRH1IDO1CYP19A1GBA1
SCHEMBL7263051 0.77 IDO1 (0.48) IDO1CYP19A1CYP2D6CYP2C19GBA1
SCHEMBL714536 0.77 HTR2A (0.52) HTR2AHRH1IDO1CYP19A1RET
SCHEMBL29593942 0.77 HTR2A (0.52) HTR2AHRH1IDO1CYP19A1RET
SCHEMBL8291564 0.76 IDO1 (0.49) HTR2AHRH1IDO1CYP19A1GBA1
SCHEMBL9838348 0.75 IDO1 (0.47) HTR2AIDO1CYP19A1HTR2CCYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2221296-B1 FUSED INDANE COMPOUND ASTELLAS PHARMA INC (JP) 2012-09-05 EP disclosed
EP-0690843-B1 Formyl- or cyano- substituted indole derivatives having dopaminergic activity UPJOHN CO (US) 2000-08-30 EP disclosed
US-5639778-A TREATING CENTRAL NERVOUS SYSTEM DISORDERS PHARMACIA & UPJOHN COMPANY (US) 1997-06-17 US disclosed
EP-0690843-A1 INDOLETETRALINS HAVING DOPAMINERGIC ACTIVITY PHARMACIA & UPJOHN COMPANY (US) 1996-01-10 EP disclosed
WO-1994021608-A1 INDOLETETRALINS HAVING DOPAMINERGIC ACTIVITY THE UPJOHN COMPANY (US) 1994-09-29 WO disclosed