SCHEMBL7445937

SCHEMBL7445937

CCOC(=O)CCN(C(=O)Oc1ccc2[nH]c(CCc3ccc(C(=N)N)s3)nc2c1C)c1ccccn1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NQO2 P16083 1/20 0.39
MAPT P10636 1/20 0.35
CHEK1 O14757 1/20 0.33
NR1I2 O75469 1/20 0.32
F2 P00734 1/20 0.32
ADORA3 P0DMS8 1/20 0.32
SLC6A2 P23975 1/20 0.32
AGTR1 P30556 1/20 0.32
SLC6A3 Q01959 1/20 0.32
SCN5A Q14524 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
HSD17B10 Q99714 1/20 0.32
TMPRSS15 P98073 2/20 0.32
MEN1 O00255 1/20 0.31
ALDH1A1 P00352 1/20 0.31
GAA P10253 1/20 0.31
MAPK1 P28482 1/20 0.31
KMT2A Q03164 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
F9 P00740 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7444344 0.99 NQO2 (0.39) NQO2MAPTCHEK1NR1I2F2
SCHEMBL7443847 0.93 F2 (0.34) NQO2F2TMPRSS15HDAC1BRD4
Hydrochloric Acid SCHEMBL7445405 0.86 NQO2 (0.45) NQO2MAPTCHEK1NR1I2F2
Hydrochloric Acid SCHEMBL7454240 0.85 NQO2 (0.40) NQO2MAPTCHEK1NR1I2F2
Hydrochloric Acid SCHEMBL7447095 0.82 NQO2 (0.54) NQO2MAPTNR1I2F2ADORA3
Hydrochloric Acid SCHEMBL7445265 0.81 NQO2 (0.44) NQO2MAPTCHEK1NR1I2F2
SCHEMBL7454396 0.81 NQO2 (0.38) NQO2MAPTNR1I2F2ADORA3
Hydrochloric Acid SCHEMBL7447918 0.80 NQO2 (0.45) NQO2MAPTCHEK1NR1I2F2
Hydrochloric Acid SCHEMBL7448525 0.80 NQO2 (0.41) NQO2MAPTCHEK1NR1I2F2
SCHEMBL7445932 0.80 F2 (0.41) NQO2F2TMPRSS15BRD4CREBBP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0966454-A1 DISUBSTITUTED BICYCLIC HETEROCYCLES, THEIR PRODUCTION AND USE AS MEDICAMENTS Boehringer Ingelheim Pharma KG (DE) 1999-12-29 EP disclosed
WO-1998037075-A1 DISUBSTITUTED BICYCLIC HETEROCYCLES, THEIR PRODUCTION AND USE AS MEDICAMENTS BOEHRINGER INGELHEIM PHARMA KG (DE) 1998-08-27 WO disclosed