SCHEMBL7446136

SCHEMBL7446136

Cc1ccc(S(=O)(=O)N2CCC[C@H]2C(=O)N[C@@H](Cc2ccc(NC(=O)CCCN)cc2)C(=O)O)cc1.Cc1ccc(S(=O)(=O)N2CCC[C@H]2C(=O)N[C@@H](Cc2ccc(NC(=O)CCCNC(=O)OC(C)(C)C)cc2)C(=O)O)cc1

nearest known ligand 0.65

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 15/20 0.65
ITGA5 P08648 5/20 0.65
ITGAV P06756 11/20 0.60
ITGA4 P13612 2/20 0.52
CA1 P00915 1/20 0.47
CA2 P00918 1/20 0.47
ITGB3 P05106 1/20 0.47
FKBP1A P62942 1/20 0.46
TSHR P16473 1/20 0.43
MAPK1 P28482 1/20 0.43
PLAU P00749 1/20 0.43
HPN P05981 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7325049 0.97 ITGB1 (0.63) ITGB1ITGA5ITGAVITGA4CA1
SCHEMBL7319362 0.90 ITGB1 (0.79) ITGB1ITGA5ITGAVITGA4ITGB3
SCHEMBL7317563 0.88 ITGB1 (0.63) ITGB1ITGA5ITGAVITGA4TSHR
SCHEMBL7327703 0.85 ITGB1 (0.70) ITGB1ITGA5ITGAVITGA4FKBP1A
SCHEMBL7325692 0.85 ITGB1 (0.61) ITGB1ITGA5ITGAVITGA4TSHR
SCHEMBL18348970 0.84 ITGB1 (0.67) ITGB1ITGA5ITGAVITGA4ITGB3
SCHEMBL7448876 0.84 ITGB1 (0.57) ITGB1ITGA5ITGAVITGA4TSHR
SCHEMBL18349161 0.84 ITGB1 (0.92) ITGB1ITGA5ITGAVITGA4ITGB3
SCHEMBL18339179 0.84 ITGB1 (0.92) ITGB1ITGA5ITGAVITGA4ITGB3
SCHEMBL16598570 0.84 ITGB1 (0.92) ITGB1ITGA5ITGAVITGA4ITGB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1001972-A1 SUBSTITUTED PHENYLALANINE TYPE COMPOUNDS WHICH INHIBIT LEUKOCYTE ADHESION MEDIATED BY VLA-4 Elan Pharmaceuticals, Inc. (US) 2000-05-24 EP claimed
WO-1999006431-A1 SUBSTITUTED PHENYLALANINE TYPE COMPOUNDS WHICH INHIBIT LEUKOCYTE ADHESION MEDIATED BY VLA-4 ELAN PHARMACEUTICALS, INC. (US) 1999-02-11 WO claimed