SCHEMBL7447328

SCHEMBL7447328

O=C(O)C1CCN(c2nc(NCc3ccc4occc4c3)c3cc(Cl)ccc3n2)CC1

nearest known ligand 0.72

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 2/20 0.72
PDE4B Q07343 2/20 0.72
PDE4C Q08493 2/20 0.72
PDE4D Q08499 2/20 0.72
PDE2A O00408 1/20 0.62
PDE5A O76074 1/20 0.62
PDE1A P54750 1/20 0.62
PDE1B Q01064 1/20 0.62
PDE1C Q14123 1/20 0.62
HRH4 Q9H3N8 16/20 0.53
HTR3A P46098 4/20 0.52
HRH1 P35367 2/20 0.52
CTNNB1 P35222 2/20 0.46
TCF7L2 Q9NQB0 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7129772 0.90 PDE4A (0.58) PDE4APDE4BPDE4CPDE4DPDE2A
SCHEMBL7499338 0.85 PDE4A (0.75) PDE4APDE4BPDE4CPDE4DPDE2A
SCHEMBL149748 0.83 PDE4A (1.00) PDE4APDE4BPDE4CPDE4DPDE2A
SCHEMBL5917665 0.83 PDE4A (0.98) PDE4APDE4BPDE4CPDE4DPDE2A
Hydrochloric Acid SCHEMBL7502602 0.83 PDE4A (0.98) PDE4APDE4BPDE4CPDE4DPDE2A
SCHEMBL5917668 0.83 PDE4A (0.98) PDE4APDE4BPDE4CPDE4DPDE2A
Potassium SCHEMBL7504150 0.83 PDE4A (0.98) PDE4APDE4BPDE4CPDE4DPDE2A
SCHEMBL7504141 0.83 PDE4A (0.98) PDE4APDE4BPDE4CPDE4DPDE2A
Hydrochloric Acid SCHEMBL29801523 0.83 PDE4A (0.98) PDE4APDE4BPDE4CPDE4DPDE2A
SCHEMBL7794280 0.83 PDE4A (0.71) PDE4APDE4BPDE4CPDE4DPDE2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0941086-A4 NITROSATED AND NITROSYLATED PHOSPHODIESTERASE INHIBITOR COMPOUNDS, COMPOSITIONS AND THEIR USES NITROMED INC (US) 2000-07-12 EP disclosed
EP-0941086-A1 NITROSATED AND NITROSYLATED PHOSPHODIESTERASE INHIBITOR COMPOUNDS, COMPOSITIONS AND THEIR USES Nitromed, Inc. (US) 1999-09-15 EP disclosed
WO-1998019672-A9 NITROSATED AND NITROSYLATED PHOSPHODIESTERASE INHIBITOR COMPOUNDS, COMPOSITIONS AND THEIR USES 1998-09-11 WO disclosed
WO-1998019672-A1 NITROSATED AND NITROSYLATED PHOSPHODIESTERASE INHIBITOR COMPOUNDS, COMPOSITIONS AND THEIR USES NITROMED INC. (US) 1998-05-14 WO disclosed