SCHEMBL7447463

SCHEMBL7447463

Cn1c(CNc2ccc(C#N)cc2)nc2ccccc21

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 15/20 0.72
RAB9A P51151 15/20 0.72
SMN1; SMN2 Q16637 9/20 0.72
KDM4E B2RXH2 4/20 0.72
TP53 P04637 4/20 0.71
ALDH1A1 P00352 4/20 0.71
L3MBTL1 Q9Y468 3/20 0.71
NFKB1 P19838 2/20 0.71
NFKB2 Q00653 2/20 0.71
RELA Q04206 2/20 0.71
ALOX15 P16050 1/20 0.71
LMNA P02545 5/20 0.70
MAPT P10636 5/20 0.70
KMT2A Q03164 3/20 0.70
MEN1 O00255 2/20 0.70
GFER P55789 2/20 0.70
MAPK1 P28482 1/20 0.70
GAA P10253 4/20 0.63
KLK1 P06870 1/20 0.62
KLK5 Q9Y337 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6779729 0.91 NPC1 (0.60) NPC1RAB9ASMN1; SMN2KDM4ETP53
SCHEMBL31243047 0.84 NPC1 (1.00) NPC1RAB9ASMN1; SMN2KDM4ETP53
SCHEMBL7415015 0.84 NPC1 (0.61) NPC1RAB9ASMN1; SMN2KDM4ETP53
SCHEMBL16268668 0.84 NPC1 (0.50) NPC1RAB9ASMN1; SMN2KDM4ETP53
SCHEMBL14914339 0.83 HDAC6 (0.51) NPC1RAB9ASMN1; SMN2KDM4ETP53
SCHEMBL2245500 0.82 NPC1 (1.00) NPC1RAB9ASMN1; SMN2KDM4ETP53
SCHEMBL13779307 0.82 NPC1 (1.00) NPC1RAB9ASMN1; SMN2KDM4ETP53
SCHEMBL2250039 0.81 NPC1 (0.77) NPC1RAB9ASMN1; SMN2KDM4ETP53
SCHEMBL19339630 0.80 HDAC6 (0.48) NPC1RAB9ASMN1; SMN2KDM4ETP53
SCHEMBL6634815 0.80 NPC1 (0.52) NPC1RAB9ASMN1; SMN2KDM4ETP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0966454-A1 DISUBSTITUTED BICYCLIC HETEROCYCLES, THEIR PRODUCTION AND USE AS MEDICAMENTS Boehringer Ingelheim Pharma KG (DE) 1999-12-29 EP disclosed
WO-1998037075-A1 DISUBSTITUTED BICYCLIC HETEROCYCLES, THEIR PRODUCTION AND USE AS MEDICAMENTS BOEHRINGER INGELHEIM PHARMA KG (DE) 1998-08-27 WO disclosed