SCHEMBL7447741

SCHEMBL7447741

CCCCCc1c(SC)nc(N)nc1-c1ccco1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 4/20 0.46
KDM4E B2RXH2 3/20 0.46
NPSR1 Q6W5P4 2/20 0.46
ADORA2A P29274 14/20 0.43
ADORA1 P30542 9/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
MEN1 O00255 2/20 0.40
ALDH1A1 P00352 2/20 0.40
POLB P06746 2/20 0.40
MAPT P10636 2/20 0.40
ALOX15 P16050 2/20 0.40
PTPN7 P35236 2/20 0.40
RECQL P46063 2/20 0.40
BLM P54132 2/20 0.40
KMT2A Q03164 2/20 0.40
HSD17B10 Q99714 2/20 0.40
TDP1 Q9NUW8 2/20 0.40
PDE4B Q07343 1/20 0.40
GAPDH P04406 1/20 0.40
NR4A1 P22736 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7146733 0.86 ADORA2A (0.47) HPGDKDM4ENPSR1ADORA2AADORA1
SCHEMBL21313152 0.84 ADORA2A (0.51) HPGDKDM4ENPSR1ADORA2AADORA1
SCHEMBL7396653 0.79 ADORA2A (0.43) HPGDKDM4ENPSR1ADORA2AADORA1
SCHEMBL7146915 0.79 ADORA2A (0.51) HPGDKDM4ENPSR1ADORA2AADORA1
SCHEMBL16229314 0.79 HPGD (0.48) HPGDKDM4ENPSR1ADORA2AADORA1
SCHEMBL12495836 0.79 ADORA2A (0.55) HPGDKDM4ENPSR1ADORA2AADORA1
SCHEMBL7146794 0.78 ADORA2A (0.49) HPGDKDM4ENPSR1ADORA2AADORA1
SCHEMBL12496524 0.77 HPGD (0.47) HPGDKDM4ENPSR1ADORA2AADORA1
SCHEMBL12496017 0.76 ADORA2A (0.58) HPGDKDM4ENPSR1ADORA2AADORA1
SCHEMBL21313215 0.76 ADORA2A (0.47) HPGDKDM4ENPSR1ADORA2AADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1261327-A2 ADENOSINE RECEPTOR MODULATORS F.HOFFMANN-LA ROCHE AG (CH) 2002-12-04 EP disclosed
WO-2001062233-A2 ADENOSINE RECEPTOR MODULATORS F. HOFFMANN LA ROCHE AG (CH) 2001-08-30 WO disclosed