SCHEMBL7448269

SCHEMBL7448269

N[C@@H](Cc1ccccc1)C(=O)N(F)[C@@H](Cc1ccc(F)cc1)C(=O)O

nearest known ligand 0.51

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SLC7A5 Q01650 3/20 0.51
ALPI P09923 1/20 0.51
PKM P14618 1/20 0.51
PTGS1 P23219 1/20 0.51
XIAP P98170 1/20 0.51
PPARG P37231 1/20 0.45
PPARA Q07869 1/20 0.45
MC4R P32245 2/20 0.43
MC3R P41968 2/20 0.43
ALDH1A1 P00352 1/20 0.43
TPH1 P17752 2/20 0.43
SLC1A3 P43003 2/20 0.42
SLC1A2 P43004 2/20 0.42
SLC1A1 P43005 2/20 0.42
SLC15A1 P46059 1/20 0.42
KIF11 P52732 2/20 0.41
MC5R P33032 1/20 0.41
LTA4H P09960 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7445543 0.85 SLC7A5 (0.50) SLC7A5ALPIPKMPTGS1XIAP
SCHEMBL7448659 0.82 SLC7A5 (0.47) SLC7A5ALPIPKMPTGS1XIAP
SCHEMBL7453774 0.81 SLC7A5 (0.46) SLC7A5ALPIPKMPTGS1XIAP
SCHEMBL28222736 0.81 ANPEP (0.54) SLC7A5ALPIPKMPTGS1XIAP
SCHEMBL8016051 0.81 ANPEP (0.54) SLC7A5ALPIPKMPTGS1XIAP
Phenylalanine SCHEMBL7525344 0.81 SLC7A5 (0.79) SLC7A5ALPIPKMPTGS1XIAP
Dl-Phenylalanine SCHEMBL7525343 0.81 SLC7A5 (0.79) SLC7A5ALPIPKMPTGS1XIAP
SCHEMBL10584413 0.78 SLC7A5 (0.62) SLC7A5ALPIPKMPTGS1XIAP
SCHEMBL7531787 0.76 ALPI (0.50) SLC7A5ALPIPKMPTGS1XIAP
SCHEMBL7531784 0.76 ALPI (0.50) SLC7A5ALPIPKMPTGS1XIAP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6221888-B1 ANTIHISTAMINE, ANTIINFLAMMATORY AGENT, AUTOIMMUNE DISEASE, RHEUMATIC DISORDERS MERCK & CO., INC. 2001-04-24 US disclosed
EP-0998282-A4 SULFONAMIDES AS CELL ADHESION INHIBITORS MERCK & CO INC (US) 2000-08-30 EP disclosed
EP-0998282-A1 SULFONAMIDES AS CELL ADHESION INHIBITORS Merck & Co., Inc. (a New Jersey corp.) (US) 2000-05-10 EP disclosed
WO-1998053818-A1 SULFONAMIDES AS CELL ADHESION INHIBITORS MERCK & CO., INC. (US) 1998-12-03 WO disclosed