SCHEMBL7448461

SCHEMBL7448461

CCCCOC(=O)NC(=N)c1ccc(N(C)Cc2nc3c(C)c(OC(=O)N(CCC(=O)OCC)c4ccccn4)ccc3[nH]2)cc1

nearest known ligand 0.35

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NQO2 P16083 1/20 0.35
NR1I2 O75469 1/20 0.35
F2 P00734 1/20 0.35
ADORA3 P0DMS8 1/20 0.35
SLC6A2 P23975 1/20 0.35
AGTR1 P30556 1/20 0.35
SLC6A3 Q01959 1/20 0.35
SCN5A Q14524 1/20 0.35
ALDH1A1 P00352 2/20 0.32
MEN1 O00255 1/20 0.32
GAA P10253 1/20 0.32
MAPK1 P28482 1/20 0.32
KMT2A Q03164 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
HDAC6 Q9UBN7 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.30
HSD17B10 Q99714 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7452917 0.98 NR1I2 (0.38) NQO2NR1I2F2ADORA3SLC6A2
SCHEMBL7448886 0.98 NR1I2 (0.38) NQO2NR1I2F2ADORA3SLC6A2
SCHEMBL7454126 0.90 NQO2 (0.37) NQO2NR1I2F2ADORA3SLC6A2
Hydrochloric Acid SCHEMBL7445265 0.88 NQO2 (0.44) NQO2NR1I2F2ADORA3SLC6A2
SCHEMBL7451787 0.88 NR1I2 (0.39) NQO2NR1I2F2ADORA3SLC6A2
SCHEMBL7453707 0.87 F2 (0.46) NQO2NR1I2F2ADORA3SLC6A2
SCHEMBL5555934 0.87 F2 (0.46) NQO2NR1I2F2ADORA3SLC6A2
SCHEMBL7453308 0.86 NQO2 (0.40) NQO2NR1I2F2ADORA3SLC6A2
SCHEMBL7446902 0.84 F2 (0.41) NQO2NR1I2F2ADORA3SLC6A2
SCHEMBL7452514 0.83 F2 (0.42) NQO2NR1I2F2ADORA3SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0966454-A1 DISUBSTITUTED BICYCLIC HETEROCYCLES, THEIR PRODUCTION AND USE AS MEDICAMENTS Boehringer Ingelheim Pharma KG (DE) 1999-12-29 EP disclosed
WO-1998037075-A1 DISUBSTITUTED BICYCLIC HETEROCYCLES, THEIR PRODUCTION AND USE AS MEDICAMENTS BOEHRINGER INGELHEIM PHARMA KG (DE) 1998-08-27 WO disclosed