SCHEMBL7451202

SCHEMBL7451202

N#CC1(c2ccc(OC(F)F)c(OCC3CC3)c2)CCC(C(=O)O)CC1.[Fe]

nearest known ligand 0.58

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 20/20 0.58
PDE4A P27815 16/20 0.58
PDE4C Q08493 16/20 0.58
PDE4D Q08499 16/20 0.58
ABCB11 O95342 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6197797 0.99 PDE4B (0.59) PDE4BPDE4APDE4CPDE4DABCB11
SCHEMBL6196611 0.99 PDE4B (0.59) PDE4BPDE4APDE4CPDE4DABCB11
SCHEMBL6196613 0.99 PDE4B (0.59) PDE4BPDE4APDE4CPDE4DABCB11
SCHEMBL7451195 0.89 PDE4B (0.50) PDE4BPDE4APDE4CPDE4DABCB11
SCHEMBL6196516 0.89 PDE4B (0.63) PDE4BPDE4APDE4CPDE4D
SCHEMBL6545778 0.89 PDE4B (0.63) PDE4BPDE4APDE4CPDE4D
SCHEMBL6196511 0.89 PDE4B (0.63) PDE4BPDE4APDE4CPDE4D
SCHEMBL6199802 0.89 PDE4B (0.55) PDE4BPDE4APDE4CPDE4DABCB11
SCHEMBL6197472 0.89 PDE4B (0.55) PDE4BPDE4APDE4CPDE4DABCB11
SCHEMBL5799817 0.89 PDE4B (0.55) PDE4BPDE4APDE4CPDE4DABCB11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1043994-A4 METHOD FOR TREATING MULTIPLE SCLEROSIS SMITHKLINE BEECHAM CORP (US) 2002-09-11 EP claimed
EP-1043994-A1 METHOD FOR TREATING MULTIPLE SCLEROSIS SMITHKLINE BEECHAM CORPORATION (US) 2000-10-18 EP claimed
WO-1999034797-A1 METHOD FOR TREATING MULTIPLE SCLEROSIS SMITHKLINE BEECHAM CORPORATION (US) 1999-07-15 WO claimed