SCHEMBL7454096

SCHEMBL7454096

O=C(O)[C@H]1CCCC[C@H]1Cc1cccnc1

nearest known ligand 0.49

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NAPRT Q6XQN6 1/20 0.47
KDM4E B2RXH2 3/20 0.47
POLB P06746 1/20 0.47
ALDH1A1 P00352 2/20 0.44
PKM P14618 1/20 0.44
TSHR P16473 1/20 0.43
CHRNA7 P36544 4/20 0.43
CHRNB2 P17787 2/20 0.43
CHRNA4 P43681 2/20 0.43
TBXAS1 P24557 2/20 0.42
HSD17B10 Q99714 1/20 0.42
TAAR1 Q96RJ0 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7454090 1.00 NAPRT (0.47) NAPRTKDM4EPOLBALDH1A1PKM
SCHEMBL7225398 1.00 NAPRT (0.47) NAPRTKDM4EPOLBALDH1A1PKM
SCHEMBL7230439 0.83 TAAR1 (0.53) KDM4EPOLBALDH1A1TAAR1
SCHEMBL7452644 0.83 TAAR1 (0.53) KDM4EPOLBALDH1A1TAAR1
SCHEMBL7452648 0.83 TAAR1 (0.53) KDM4EPOLBALDH1A1TAAR1
SCHEMBL5002695 0.82 HSD17B10 (0.56) KDM4EALDH1A1HSD17B10TAAR1
SCHEMBL7223358 0.82 HSD17B10 (0.56) KDM4EALDH1A1HSD17B10TAAR1
SCHEMBL1818892 0.76 NAPRT (0.46) NAPRTKDM4EPOLBALDH1A1TSHR
SCHEMBL11404025 0.75 HSD17B10 (0.37) NAPRTKDM4ETSHRHSD17B10
SCHEMBL23235646 0.73 GRM2 (0.44) TSHRHSD17B10TAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1161416-A1 ALPHA-AMINOACETIC ACID DERIVATIVES USEFUL AS ALPHA 4 BETA 7 - RECEPTOR ANTAGONISTS Elan Pharmaceuticals, Inc. (US) 2001-12-12 EP disclosed
WO-2000051974-A1 ALPHA-AMINOACETIC ACID DERIVATIVES USEFUL AS ALPHA 4 BETA 7 - RECEPTOR ANTAGONISTS ELAN PHARMACEUTICALS, INC. (US) 2000-09-08 WO disclosed