SCHEMBL7455147

SCHEMBL7455147

ClCCCc1ccnc(Cl)c1

nearest known ligand 0.59

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
RECQL P46063 1/20 0.59
LOX P28300 1/20 0.59
LOXL3 P58215 1/20 0.59
LOXL2 Q9Y4K0 1/20 0.59
GSK3A P49840 4/20 0.41
GSK3B P49841 4/20 0.41
GRM5 P41594 1/20 0.40
FFAR1 O14842 1/20 0.36
TRPA1 O75762 1/20 0.36
EPHX1 P07099 1/20 0.35
MGMT P16455 1/20 0.34
IDO1 P14902 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
SMARCA2 P51531 1/20 0.33
SMARCA4 P51532 1/20 0.33
IGF1R P08069 1/20 0.32
ALOX15 P16050 1/20 0.32
GHSR Q92847 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24668667 0.84 RECQL (0.55) RECQLLOXLOXL3LOXL2GSK3A
SCHEMBL23152494 0.84 RECQL (0.66) RECQLLOXLOXL3LOXL2GSK3A
SCHEMBL4074777 0.82 RECQL (0.53) RECQLLOXLOXL3LOXL2GSK3A
SCHEMBL27902689 0.81 RECQL (0.52) RECQLLOXLOXL3LOXL2TDP1
SCHEMBL27878725 0.81 RECQL (0.52) RECQLLOXLOXL3LOXL2TDP1
Hydrochloric Acid SCHEMBL28861654 0.81 LOX (0.61) RECQLLOXLOXL3LOXL2GSK3A
SCHEMBL27672336 0.81 RECQL (0.52) RECQLLOXLOXL3LOXL2TDP1
SCHEMBL1503624 0.80
Hydrochloric Acid SCHEMBL28231152 0.80 LOX (0.59) RECQLLOXLOXL3LOXL2GSK3A
Hydrochloric Acid SCHEMBL28232181 0.80 LOX (0.59) RECQLLOXLOXL3LOXL2GSK3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6362336-B1 ADMINISTERING A QUINAZOLINE DERIVATIVE TO A WARM-BLOODED ANIMAL FOR PRODUCING AN ANTIANGIOGENIC AND/OR VASCULAR PERMEABILITY REDUCING EFFECT ZENECA LIMITED (GB) 2002-03-26 US disclosed
US-20020032208-A1 Chemical compounds ZENECA LIMITED 2002-03-14 US disclosed
EP-0873319-B1 QUINAZOLINE DERIVATIVES ASTRAZENECA AB (SE) 2001-07-25 EP disclosed
US-6258951-B1 ANTICANCER, ANTIARTHRITIC AGENTS ZENECA LIMITED (GB) 2001-07-10 US disclosed
US-6071921-A Chemical compounds ZENECA LIMITED (GB) 2000-06-06 US disclosed
US-5962458-A ANGIOGENESIS INHIBITORS, ANTICANCER AGENTS, ANTIDIABETIC AGENTS, SKIN DISORDERS, AUTOIMMUNE DISEASES, ANTIINFLAMMATORY AGENTS, VISION DEFECTS ZENECA LIMITED (GB) 1999-10-05 US disclosed
EP-0873319-A1 QUINAZOLINE DERIVATIVES ZENECA LIMITED (GB) 1998-10-28 EP disclosed
WO-1997022596-A1 QUINAZOLINE DERIVATIVES ZENECA LIMITED (GB) 1997-06-26 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020032208-A1 Chemical compounds FLT1, CNKSR1, KDR RECQL 1574/4885LOX 1018/4885LOXL3 2422/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.