SCHEMBL7455263

SCHEMBL7455263

CCCN(O)C(=O)C(C)NC(=O)OC(C)(C)C

nearest known ligand 0.49

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.45
CA7 P43166 2/20 0.45
CA12 O43570 1/20 0.45
CA14 Q9ULX7 1/20 0.45
CA2 P00918 1/20 0.44
CTSK P43235 11/20 0.43
CYP2D6 P10635 1/20 0.40
CTSS P25774 5/20 0.40
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14737623 0.87 CA1 (0.46) CA1CA7CA2CTSKCYP2D6
SCHEMBL5447582 0.79 CA1 (0.47) CA1CA7CA2CTSKCYP2D6
SCHEMBL14923588 0.78 CA1 (0.46) CA1CA7CA12CA14CA2
SCHEMBL12915836 0.78 CA1 (0.46) CA1CA7CA12CA14CA2
SCHEMBL16232686 0.78 CA1 (0.46) CA1CA7CA12CA14CA2
SCHEMBL5873409 0.78 CA1 (0.46) CA1CA7CA2CTSKCYP2D6
SCHEMBL5433610 0.78 CA1 (0.46) CA1CA7CA2CTSKCYP2D6
SCHEMBL6632972 0.76 CA1 (0.47) CA1CA7CA12CA14CA2
SCHEMBL768534 0.76 CA1 (0.47) CA1CA7CA12CA14CA2
SCHEMBL2386106 0.76 CA1 (0.47) CA1CA7CA12CA14CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1051176-A4 SUBSTITUTED OXOAZAHETEROCYCLYL FACTOR Xa INHIBITORS AVENTIS PHARM PROD INC (US) 2002-06-12 EP disclosed
EP-1051176-A1 SUBSTITUTED OXOAZAHETEROCYCLYL FACTOR Xa INHIBITORS Aventis Pharmaceuticals Products Inc. (US) 2000-11-15 EP disclosed
WO-1999037304-A1 SUBSTITUTED OXOAZAHETEROCYCLYL FACTOR Xa INHIBITORS AVENTIS PHARMACEUTICALS PRODUCTS INC. (US) 1999-07-29 WO disclosed