SCHEMBL7457045

SCHEMBL7457045

C[n+]1ccccc1C#N.Fc1c(F)c(F)c([B-](c2c(F)c(F)c(F)c(F)c2F)(c2c(F)c(F)c(F)c(F)c2F)c2c(F)c(F)c(C(F)(F)F)c(F)c2F)c(F)c1F

nearest known ligand 0.55

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
HDAC8 Q9BY41 2/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL577676 0.90 HDAC8 (0.68) HDAC8
SCHEMBL29815870 0.90 HDAC8 (0.68) HDAC8
SCHEMBL7459440 0.83 HDAC8 (0.57) HDAC8
SCHEMBL7457967 0.75 SLC22A2 (0.31)
SCHEMBL8988114 0.74 HDAC8 (1.00) HDAC8
SCHEMBL862249 0.74
Iodide SCHEMBL30133746 0.73 HDAC8 (0.95) HDAC8
Hydrochloric Acid SCHEMBL5833068 0.73 HDAC8 (0.95) HDAC8
SCHEMBL7460697 0.71 CHKA (0.35)
SCHEMBL577775 0.70 HDAC8 (0.75) HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0690079-B1 ETHYLENE COPOLYMER, THERMOPLASTIC RESIN COMPOSITION CONTAINING THE SAME, AND PROCESS FOR PRODUCING ETHYLENE COPOLYMER IDEMITSU KOSAN CO (JP) 2002-07-03 EP disclosed
EP-0683184-B1 POLYETHYLENE, THERMOPLASTIC RESIN COMPOSITION CONTAINING THE SAME, AND PROCESS FOR PRODUCING POLYETHYLENE IDEMITSU KOSAN CO (JP) 2002-06-12 EP disclosed
US-6169154-B1 MACROMONOMER DERIVABLE FROM ETHYLENE SINGLY OR DERIVABLE FROM ETHYLENE AND ANOTHER OLEFIN, THE MACROMONOMER HAVING A BRANCH OTHER THAN THE BRANCH DERIVED FROM THE OTHER OLEFIN; CAN BE HYDROGENATED TO PROVIDE A WAX IDEMITSU KOSAN CO., LTD. (JP) 2001-01-02 US disclosed
US-6121402-A EXCELLENT IN WORKING PROPERTIES AND PERMITS THE CONTROL OF PHYSICAL PROPERTIES SUCH AS DENSITY, A MELTING POINT AND CRYSTALLINITY MAINLY IN THE STATE OF A HOMOPOLYMER IDEMITSU KOSAN CO., LTD. (JP) 2000-09-19 US disclosed
EP-0727446-B1 BRANCHED ETHYLENE MACROMONOMER AND POLYMER PRODUCED THEREFROM IDEMITSU KOSAN CO (JP) 2000-09-13 EP disclosed
US-5955557-A Branched ethylenic macromonomer and its polymer IDEMITSU KOSAN CO., LTD. (JP) 1999-09-21 US disclosed
US-5747620-A CATALYTIC ADDITION POLYMERIZATION WITH COORDINATION CATALYSTS IDEMITSU KOSAN CO., LTD. (JP) 1998-05-05 US disclosed
EP-0690079-A1 ETHYLENE COPOLYMER, THERMOPLASTIC RESIN COMPOSITION CONTAINING THE SAME, AND PROCESS FOR PRODUCING ETHYLENE COPOLYMER IDEMITSU KOSAN COMPANY LIMITED (JP) 1996-01-03 EP disclosed
EP-0683184-A1 POLYETHYLENE, THERMOPLASTIC RESIN COMPOSITION CONTAINING THE SAME, AND PROCESS FOR PRODUCING POLYETHYLENE IDEMITSU KOSAN COMPANY LIMITED (JP) 1995-11-22 EP disclosed