SCHEMBL7459663

SCHEMBL7459663

C[C@H](O)[C@@H](CCCc1ccccc1)n1cnc2c(N)ncnc21

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ADA P00813 4/20 0.69
PDE2A O00408 3/20 0.69
CYP3A4 P08684 2/20 0.69
PDE4A P27815 1/20 0.69
PDE4B Q07343 1/20 0.69
PDE4C Q08493 1/20 0.69
PDE4D Q08499 1/20 0.69
KDM4E B2RXH2 1/20 0.69
ALDH1A1 P00352 1/20 0.69
CYP1A2 P05177 1/20 0.69
ALOX15 P16050 1/20 0.69
SMN1; SMN2 Q16637 1/20 0.69
HSD17B10 Q99714 1/20 0.69
TSHR P16473 1/20 0.69
HIF1A Q16665 1/20 0.69
LMNA P02545 1/20 0.67
BLM P54132 1/20 0.67

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7458479 0.97 ADA (0.71) ADAPDE2ACYP3A4PDE4APDE4B
SCHEMBL7458088 0.96 ADA (0.72) ADAPDE2ACYP3A4PDE4APDE4B
SCHEMBL7456900 0.93
Hydrochloric Acid SCHEMBL1740511 0.92
SCHEMBL8577504 0.86 ADA (0.65) ADAPDE2ACYP3A4PDE4APDE4B
SCHEMBL7458391 0.86 ADA (0.65) ADAPDE2ACYP3A4PDE4APDE4B
SCHEMBL7452717 0.85 ADA (0.50) ADAPDE2ACYP3A4PDE4APDE4B
SCHEMBL8585199 0.83 ADA (0.82) ADAPDE2ACYP3A4PDE4APDE4B
SCHEMBL16395274 0.83 ADA (0.67) ADAPDE2ACYP3A4PDE4APDE4B
SCHEMBL15270317 0.83 ADA (0.67) ADAPDE2ACYP3A4PDE4APDE4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0936911-B1 ADENOSINE DEAMINASE INHIBITORS RHODE ISLAND EDUCATION (US) 2002-04-10 EP disclosed
EP-0936911-A4 1999-10-06 EP disclosed
EP-0936911-A1 ADENOSINE DEAMINASE INHIBITORS THE BOARD OF GOVERNORS FOR HIGHER EDUCATION STATE OF RHODE ISLAND AND PROVIDENCE PLANTATIONS (US) 1999-08-25 EP disclosed
WO-1998002166-A1 ADENOSINE DEAMINASE INHIBITORS THE BOARD OF GOVERNORS FOR HIGHER EDUCATION, STATE OF RHODE ISLAND AND PROVIDENCE PLANTATIONS (US) 1998-01-22 WO disclosed
US-5703084-A Adenosine deaminase inhibitors THE BOARD OF GOVERNORS FOR HIGHER EDUCATION, STATE OF RHODE ISLAND AND PROVIDENCE PLANTATIONS (US) 1997-12-30 US disclosed