SCHEMBL7463194

SCHEMBL7463194

CCc1cc(C=C2SC(=O)NC2=O)ccc1-c1cc2c(cc1C(F)(F)F)C(C)(C)CCC2(C)C

nearest known ligand 0.47

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PIM1 P11309 7/20 0.47
PIM2 Q9P1W9 7/20 0.47
CISD1 Q9NZ45 2/20 0.47
TTR P02766 1/20 0.47
IGF1R P08069 1/20 0.47
HPGD P15428 2/20 0.46
FOXM1 Q08050 1/20 0.46
ESRRA P11474 8/20 0.46
CYP3A4 P08684 1/20 0.46
PTPN1 P18031 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7463186 1.00 PIM1 (0.47) PIM1PIM2CISD1TTRIGF1R
SCHEMBL5484274 0.93 FOXM1 (0.47) PIM1PIM2CISD1TTRIGF1R
SCHEMBL14492772 0.93 FOXM1 (0.47) PIM1PIM2CISD1TTRIGF1R
SCHEMBL5484278 0.93 FOXM1 (0.47) PIM1PIM2CISD1TTRIGF1R
SCHEMBL7461441 0.89 ESRRA (0.51) PIM1PIM2CISD1TTRHPGD
SCHEMBL7461440 0.89 ESRRA (0.51) PIM1PIM2CISD1TTRHPGD
SCHEMBL7466383 0.88 IGF1R (0.52) PIM1PIM2CISD1TTRIGF1R
SCHEMBL7466389 0.88 IGF1R (0.52) PIM1PIM2CISD1TTRIGF1R
SCHEMBL14492771 0.87 ESRRA (0.48) PIM1PIM2CISD1TTRHPGD
SCHEMBL5491435 0.87 ESRRA (0.48) PIM1PIM2CISD1TTRHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1214305-A1 BENZYLIDENE-THIAZOLIDINEDIONES AND ANALOGUES AND THEIR USE IN THE TREATMENT OF INFLAMMATION Maxia Pharmaceuticals, Inc. (US) 2002-06-19 EP disclosed
WO-2001016123-A1 BENZYLIDENE-THIAZOLIDINEDIONES AND ANALOGUES AND THEIR USE IN THE TREATMENT OF INFLAMMATION MAXIA PHARMACEUTICALS, INC. (US) 2001-03-08 WO disclosed