SCHEMBL7464696

SCHEMBL7464696

COc1ccc2cnc(Nc3ccc(N4CCN(C(N)C=O)CC4)cc3)nc2c1C1CCCC1

nearest known ligand 0.74

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 20/20 0.74
CCND1 P24385 20/20 0.74
CCNE1 P24864 15/20 0.71
CDK2 P24941 15/20 0.71
CDK1 P06493 12/20 0.71
CCNB1 P14635 12/20 0.71

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7475748 0.88 CDK4 (0.71) CDK4CCND1CCNE1CDK2CDK1
SCHEMBL7469611 0.87 CDK4 (0.69) CDK4CCND1CCNE1CDK2CDK1
SCHEMBL6088024 0.86 CDK4 (1.00) CDK4CCND1CCNE1CDK2CDK1
SCHEMBL7468854 0.85 CDK4 (0.73) CDK4CCND1CCNE1CDK2CDK1
SCHEMBL6087555 0.85 CDK4 (0.87) CDK4CCND1CCNE1CDK2CDK1
SCHEMBL6087349 0.85 CDK4 (1.00) CDK4CCND1CCNE1CDK2CDK1
SCHEMBL7461957 0.85 CDK4 (0.77) CDK4CCND1CCNE1CDK2CDK1
SCHEMBL7471048 0.84 CDK4 (0.68) CDK4CCND1CCNE1CDK2CDK1
SCHEMBL6089142 0.84 CDK4 (0.80) CDK4CCND1CCNE1CDK2CDK1
SCHEMBL7475822 0.83 CDK4 (0.74) CDK4CCND1CCNE1CDK2CDK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1235815-A1 QUINAZOLINES AND THEIR USE FOR INHIBITING CYCLIN-DEPENDENT KINASE ENZYMES WARNER-LAMBERT COMPANY (US) 2002-09-04 EP disclosed
WO-2001038315-A1 QUINAZOLINES AND THEIR USE FOR INHIBITING CYCLIN-DEPENDENT KINASE ENZYMES WARNER-LAMBERT COMPANY (US) 2001-05-31 WO disclosed