SCHEMBL7464874

SCHEMBL7464874

COC(=O)c1c(Cc2c(F)cccc2F)ccc2[nH]c(-c3c(F)cccc3F)nc12

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 11/20 0.41
PKN1 Q16512 1/20 0.40
PKN2 Q16513 1/20 0.40
BDKRB1 P46663 2/20 0.39
GRIN2B Q13224 1/20 0.36
PARP1 P09874 1/20 0.36
PTGDR2 Q9Y5Y4 2/20 0.36
MGAM O43451 1/20 0.34
GAA P10253 1/20 0.34
SI P14410 1/20 0.34
MGAM2 Q2M2H8 1/20 0.34
HPSE Q9Y251 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7472922 0.85 DHODH (0.41) DHODHPKN1PKN2GRIN2BPARP1
SCHEMBL7467113 0.83 DHODH (0.38) DHODHGRIN2BPARP1PTGDR2MGAM
SCHEMBL7474192 0.81 MGAM (0.38) DHODHGRIN2BPARP1PTGDR2MGAM
SCHEMBL7465091 0.80 DHODH (0.41) DHODHGRIN2BPARP1PTGDR2
SCHEMBL7462889 0.80 DHODH (0.41) DHODHGRIN2BPARP1PTGDR2MGAM
SCHEMBL7460756 0.80 GRIN2B (0.41) DHODHGRIN2BMGAMGAASI
SCHEMBL7469303 0.79 MGAM (0.43) DHODHGRIN2BPTGDR2MGAMGAA
SCHEMBL7463314 0.78 GRIN2B (0.41) DHODHGRIN2BPTGDR2MGAMGAA
SCHEMBL7466323 0.78 DHODH (0.41) DHODHGRIN2BPARP1MGAMGAA
SCHEMBL7468106 0.77 DHODH (0.40) DHODHGRIN2BPARP1PTGDR2MGAM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1210336-A1 SUBSTITUTED BENZIMIDAZOLES AS NON-NUCLEOSIDE INHIBITORS OF REVERSE TRANSCRIPTASE THE UNITED STATES OF AMERICA, as represented by the Secretary of the Department of Health and Human Services (US) 2002-06-05 EP disclosed
WO-2001014343-A1 SUBSTITUTED BENZIMIDAZOLES AS NON-NUCLEOSIDE INHIBITORS OF REVERSE TRANSCRIPTASE THE GOVERNMENT OF THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2001-03-01 WO disclosed