SCHEMBL7467410

SCHEMBL7467410

O=C(c1cc(C(F)(F)F)cc(C(F)(F)F)c1)N1CCN(CC#CCN2CCSCC2)C[C@H]1Cc1ccc2ccccc2c1

nearest known ligand 0.47

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 18/20 0.47
CA1 P00915 2/20 0.38
CA2 P00918 2/20 0.38
CA4 P22748 2/20 0.38
CA9 Q16790 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7555292 0.99 TACR1 (0.46) TACR1CA1CA2CA4CA9
SCHEMBL7463549 0.90 TACR1 (0.51) TACR1
Hydrochloric Acid SCHEMBL7465655 0.90 TACR1 (0.51) TACR1
SCHEMBL6133052 0.90 TACR1 (0.47) TACR1CA1CA2CA4CA9
Hydrochloric Acid SCHEMBL7463514 0.89 TACR1 (0.50) TACR1
Hydrochloric Acid SCHEMBL7472932 0.89 TACR1 (0.46) TACR1CA1CA2CA4CA9
Hydrochloric Acid SCHEMBL7460930 0.88 TACR1 (0.50) TACR1
Hydrochloric Acid SCHEMBL7460904 0.88 TACR1 (0.46) TACR1CA1CA2CA4CA9
Hydrochloric Acid SCHEMBL7460897 0.88 TACR1 (0.46) TACR1CA1CA2CA4CA9
Hydrochloric Acid SCHEMBL7467254 0.87 TACR1 (0.45) TACR1CA1CA2CA4CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0873320-B1 PIPERAZINE DERIVATIVES AS TACHYKININ ANTAGONISTS FUJISAWA PHARMACEUTICAL CO (JP) 2002-06-12 EP disclosed