SCHEMBL7469825

SCHEMBL7469825

O=C(O)c1ccc(N2CCC[C@H](Nc3ncccn3)C2)c(F)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
NPSR1 Q6W5P4 2/20 0.41
KDM4E B2RXH2 1/20 0.41
CCNK O75909 2/20 0.41
CCNA2 P20248 2/20 0.41
CDK2 P24941 2/20 0.41
CDK7 P50613 2/20 0.41
CCNH P51946 2/20 0.41
CDK12 Q9NYV4 2/20 0.41
CCNT1 O60563 1/20 0.41
CDK9 P50750 1/20 0.41
CDK13 Q14004 1/20 0.41
MAPT P10636 4/20 0.40
HPGD P15428 4/20 0.40
ALDH1A1 P00352 3/20 0.40
TSHR P16473 2/20 0.40
ROCK2 O75116 1/20 0.39
ROCK1 Q13464 1/20 0.39
CDC42BPB Q9Y5S2 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7462642 1.00 MEN1 (0.41) MEN1KMT2ANPSR1KDM4ECCNK
SCHEMBL7468744 0.89 CYP1A2 (0.43) NPSR1KDM4ECCNKCCNA2CDK2
SCHEMBL7475340 0.89 CYP1A2 (0.43) NPSR1KDM4ECCNKCCNA2CDK2
SCHEMBL7468836 0.88 EPHX2 (0.41) MEN1KMT2AKDM4ECCNKCCNA2
SCHEMBL382771 0.87 GAA (0.46) MEN1KMT2ANPSR1KDM4EMAPT
SCHEMBL7053339 0.82 CASR (0.54) MEN1KMT2ANPSR1KDM4ECASR
SCHEMBL7463214 0.82 CASR (0.54) MEN1KMT2ANPSR1KDM4ECASR
SCHEMBL7469473 0.82 MAPK8 (0.39) MEN1KMT2ANPSR1KDM4ECCNK
SCHEMBL6497606 0.81 KDM4E (0.54) MEN1KMT2AKDM4ECCNKCDK12
SCHEMBL6498986 0.81 KDM4E (0.54) MEN1KMT2AKDM4ECCNKCDK12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1227083-A1 3-AMINOPIPERIDINE DERIVATIVES AS INTEGRIN $g(a)v$g(b)3 ANTAGONISTS MEIJI SEIKA KAISHA LTD. (JP) 2002-07-31 EP disclosed