SCHEMBL7472412

SCHEMBL7472412

CCCn1c(=O)c2nc(C34CCC(CC3)CC4)[nH]c2n(CCC)c1=O

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 16/20 0.51
ADORA2A P29274 13/20 0.51
ADORA2B P29275 8/20 0.51
ADORA3 P0DMS8 4/20 0.45
SLC6A3 Q01959 1/20 0.43
SLC22A6 Q4U2R8 1/20 0.43
SLC22A8 Q8TCC7 1/20 0.43
SLC22A11 Q9NSA0 1/20 0.43
MEN1 O00255 1/20 0.43
GMNN O75496 1/20 0.43
LMNA P02545 1/20 0.43
CYP1A2 P05177 1/20 0.43
TSHR P16473 1/20 0.43
PMP22 Q01453 1/20 0.43
KMT2A Q03164 1/20 0.43
HIF1A Q16665 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1565645 0.84 ADORA1 (0.70) ADORA1ADORA2AADORA2BADORA3
SCHEMBL1566016 0.83 ADORA1 (0.50) ADORA1ADORA2AADORA2BADORA3
SCHEMBL1566166 0.83 ADORA1 (0.56) ADORA1ADORA2AADORA2BADORA3
SCHEMBL1566445 0.82 ADORA1 (0.53) ADORA1ADORA2AADORA2BADORA3
SCHEMBL1566656 0.82 ADORA1 (0.58) ADORA1ADORA2AADORA2BADORA3
SCHEMBL1567199 0.82 ADORA1 (0.58) ADORA1ADORA2AADORA2BADORA3
SCHEMBL1565447 0.81 ADORA1 (0.52) ADORA1ADORA2AADORA2BADORA3
SCHEMBL1565446 0.81 ADORA1 (0.52) ADORA1ADORA2AADORA2BADORA3
SCHEMBL7473253 0.81 ADORA1 (0.76) ADORA1ADORA2AADORA2BADORA3SLC6A3
SCHEMBL1566176 0.81 ADORA1 (0.53) ADORA1ADORA2AADORA2BADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1230243-A1 POYCYLOALKYLPURINES AS ADENOSINE RECEPTOR ANTAGONISTS BIOGEN, INC. (US) 2002-08-14 EP disclosed
WO-2001034610-A1 POLYCYCLOALKYLPURINES AS ADENOSINE RECEPTOR ANTAGONISTS BIOGEN, INC. (US) 2001-05-17 WO disclosed