SCHEMBL7472789

SCHEMBL7472789

O=C1CN(c2ccc(C3=NOC(CNc4ccon4)C3)cc2F)CCS1

nearest known ligand 0.39

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CYP2E1 P05181 1/20 0.39
MAOA P21397 2/20 0.38
MIF P14174 15/20 0.38
PDE3B Q13370 2/20 0.34
PDE3A Q14432 2/20 0.34
MAOB P27338 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5654967 0.89 MIF (0.39) CYP2E1MAOAMIFMAOB
SCHEMBL5654974 0.89 MIF (0.39) CYP2E1MAOAMIFMAOB
SCHEMBL5654348 0.85 PDE3B (0.42) CYP2E1MAOAMIFPDE3BPDE3A
SCHEMBL5654353 0.85 PDE3B (0.42) CYP2E1MAOAMIFPDE3BPDE3A
SCHEMBL5655995 0.84 MIF (0.40) CYP2E1MAOAMIFPDE3BPDE3A
SCHEMBL5656000 0.84 MIF (0.40) CYP2E1MAOAMIFPDE3BPDE3A
SCHEMBL5654102 0.84 MIF (0.39) CYP2E1MAOAMIFPDE3BPDE3A
SCHEMBL5654108 0.84 MIF (0.39) CYP2E1MAOAMIFPDE3BPDE3A
SCHEMBL5656828 0.83 KDR (0.45) CYP2E1MAOAMIFMAOB
SCHEMBL5655616 0.82 MIF (0.38) CYP2E1MAOAMIFPDE3BPDE3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1242416-A1 SUBSTITUTED ISOXAZOLINES AND THEIR USE AS ANTIBACTERIAL AGENTS AstraZeneca AB (SE) 2002-09-25 EP claimed
WO-2001040222-A1 SUBSTITUTED ISOXAZOLINES AND THEIR USE AS ANTIBACTERIAL AGENTS ASTRAZENECA AB (SE) 2001-06-07 WO claimed