SCHEMBL7472925

SCHEMBL7472925

C[C@@H]1CNCCN1c1nccnc1OCCOc1cccnc1O

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 12/20 0.42
HTR2A P28223 9/20 0.42
HTR2B P41595 8/20 0.42
KCNH2 Q12809 1/20 0.39
HTR1A P08908 1/20 0.34
SLC6A2 P23975 1/20 0.34
BRPF1 P55201 3/20 0.34
BRD1 O95696 2/20 0.34
BRD4 O60885 1/20 0.34
BRPF3 Q9ULD4 1/20 0.34
GSK3B P49841 2/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
SSTR1 P30872 1/20 0.33
SSTR4 P31391 1/20 0.33
LATS1 O95835 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4313537 0.88 HTR2C (0.42) HTR2CHTR2AHTR2BKCNH2HTR1A
SCHEMBL2639295 0.88 HTR2C (0.42) HTR2CHTR2AHTR2BKCNH2HTR1A
SCHEMBL237951 0.88 HTR2C (0.42) HTR2CHTR2AHTR2BKCNH2HTR1A
SCHEMBL905805 0.88 HTR2C (0.42) HTR2CHTR2AHTR2BKCNH2HTR1A
SCHEMBL2639565 0.88 HTR2C (0.45) HTR2CHTR2AHTR2BKCNH2HTR1A
SCHEMBL2640227 0.88 HTR2C (0.42) HTR2CHTR2AHTR2BKCNH2HTR1A
SCHEMBL2639684 0.88 HTR2C (0.42) HTR2CHTR2AHTR2BKCNH2HTR1A
SCHEMBL4308087 0.88 HTR2C (0.45) HTR2CHTR2AHTR2BKCNH2HTR1A
SCHEMBL4316338 0.88 HTR2C (0.42) HTR2CHTR2AHTR2BKCNH2HTR1A
SCHEMBL4320049 0.86 HTR2C (0.43) HTR2CHTR2AHTR2BKCNH2HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1178973-A2 NOVEL COMPOUNDS, THEIR USE AND PREPARATION Pharmacia AB (SE) 2002-02-13 EP disclosed
WO-2000076984-A2 NOVEL COMPOUNDS, THEIR USE AND PREPARATION BIOVITRUM AB (SE) 2000-12-21 WO disclosed