SCHEMBL7472961

SCHEMBL7472961

Cc1cccc2c1nc(C1CCN(Cc3ccccc3)CC1)n2C

nearest known ligand 0.51

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NPY1R P25929 3/20 0.51
PARP1 P09874 1/20 0.50
POLB P06746 2/20 0.46
TDP1 Q9NUW8 1/20 0.46
DRD2 P14416 7/20 0.46
DRD4 P21917 5/20 0.46
DRD3 P35462 5/20 0.46
ACHE P22303 1/20 0.46
GRM2 Q14416 3/20 0.46
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
PDE10A Q9Y233 1/20 0.43
HTR3E A5X5Y0 1/20 0.43
HTR3B O95264 1/20 0.43
HTR3A P46098 1/20 0.43
HTR3D Q70Z44 1/20 0.43
HTR3C Q8WXA8 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7465623 0.94 NPY1R (0.48) NPY1RPARP1POLBTDP1DRD2
SCHEMBL5622218 0.82 PARP1 (0.76) PARP1DRD2DRD4
SCHEMBL11923730 0.82 PDE10A (0.53) PARP1PDE10AHTR3A
SCHEMBL7043510 0.80 PARP1 (0.55) PARP1POLBTDP1DRD2DRD4
SCHEMBL13777216 0.79 GRM2 (0.70) NPY1RDRD2DRD4DRD3GRM2
SCHEMBL6756278 0.78 TLR7 (0.54) PARP1POLBMEN1KMT2APDE10A
SCHEMBL5620889 0.77 PARP1 (0.71) PARP1DRD2
SCHEMBL21348799 0.76 PDE10A (0.48) PARP1PDE10AHTR3A
SCHEMBL7041082 0.75 PARP1 (0.52) PARP1DRD2DRD4MEN1KMT2A
SCHEMBL13450177 0.72 MEN1 (0.67) POLBDRD2DRD4DRD3ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1133477-A1 SUBSTITUTED BENZIMIDAZOLES AND THEIR USE AS PARP INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 2001-09-19 EP disclosed
WO-2000032579-A1 SUBSTITUTED BENZIMIDAZOLES AND THEIR USE AS PARP INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 2000-06-08 WO disclosed