SCHEMBL7473358

SCHEMBL7473358

CCOC(=O)Cc1ccc(N/C(CC)=C2/C(=O)Nc3cc(OC)c(OC)cc32)cc1

nearest known ligand 0.45

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
RET P07949 5/20 0.45
MAPT P10636 4/20 0.41
LMNA P02545 2/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
KLK7 P49862 1/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
HTT P42858 1/20 0.39
EPHX2 P34913 1/20 0.39
CHEK1 O14757 1/20 0.38
GAA P10253 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6332666 1.00 RET (0.45) RETMAPTLMNASMN1; SMN2KLK7
SCHEMBL6332672 1.00 RET (0.45) RETMAPTLMNASMN1; SMN2KLK7
SCHEMBL6329199 0.89 RET (0.47) RETMAPTEPHX2GAA
SCHEMBL7474775 0.89 RET (0.47) RETMAPTEPHX2GAA
SCHEMBL6329207 0.89 RET (0.47) RETMAPTEPHX2GAA
SCHEMBL6337231 0.88 CHEK1 (0.45) RETEPHX2CHEK1GAA
SCHEMBL6337227 0.88 CHEK1 (0.45) RETEPHX2CHEK1GAA
SCHEMBL6330792 0.88 RET (0.44) RETMEN1KMT2AEPHX2CHEK1
SCHEMBL6330783 0.88 RET (0.44) RETMEN1KMT2AEPHX2CHEK1
SCHEMBL6336093 0.86 MAPT (0.54) RETMAPTLMNASMN1; SMN2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1212318-A1 SUBSTITUTED INDOLINONES AS TYROSINE KINASE INHIBITORS Boehringer Ingelheim Pharma KG (DE) 2002-06-12 EP disclosed
WO-2001016130-A1 SUBSTITUTED INDOLINONES AS TYROSINE KINASE INHIBITORS BOEHRINGER INGELHEIM PHARMA KG (DE) 2001-03-08 WO disclosed