SCHEMBL7475322

SCHEMBL7475322

[CH2]c1ccc(CN2CCN(C(C)=O)CC2)cc1

nearest known ligand 0.76

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 2/20 0.76
MEN1 O00255 2/20 0.62
KMT2A Q03164 2/20 0.62
ATM Q13315 2/20 0.62
RORC P51449 1/20 0.57
CYP2D6 P10635 1/20 0.54
CYP1A2 P05177 1/20 0.51
CYP2C9 P11712 1/20 0.51
TSHR P16473 1/20 0.51
LTA4H P09960 1/20 0.51
L3MBTL1 Q9Y468 2/20 0.50
CHRM1 P11229 1/20 0.50
HTR2A P28223 1/20 0.50
MCHR1 Q99705 1/20 0.50
SMN1; SMN2 Q16637 2/20 0.49
POLB P06746 2/20 0.49
ALDH1A1 P00352 1/20 0.49
HTT P42858 1/20 0.49
LMNA P02545 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL321890 0.85 HRH3 (0.78) HRH3MEN1KMT2AATMRORC
SCHEMBL3239820 0.85 HRH3 (0.78) HRH3MEN1KMT2AATMRORC
SCHEMBL29056068 0.85 HRH3 (0.78) HRH3MEN1KMT2AATMRORC
SCHEMBL8122521 0.85 HRH3 (0.78) HRH3MEN1KMT2AATMRORC
Hydrochloric Acid SCHEMBL7599251 0.83 HRH3 (0.88) HRH3MEN1KMT2AATMRORC
SCHEMBL3916831 0.83 HRH3 (0.76) HRH3MEN1KMT2AATMRORC
SCHEMBL1927730 0.83 HRH3 (0.76) HRH3MEN1KMT2AATMRORC
SCHEMBL1481137 0.83 HRH3 (0.76) HRH3MEN1KMT2AATMRORC
SCHEMBL1943497 0.83 HRH3 (0.75) HRH3MEN1KMT2AATMCYP2D6
Water SCHEMBL27786097 0.82 HRH3 (0.73) HRH3MEN1KMT2AATMRORC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1189609-A4 CXCR-4 RECEPTOR ANTAGONISTS - THROMBOPOIETIN MIMETICS SMITHKLINE BEECHAM CORP (US) 2002-10-30 EP disclosed
EP-1189609-A1 CXCR-4 RECEPTOR ANTAGONISTS - THROMBOPOIETIN MIMETICS SMITHKLINE BEECHAM CORPORATION (US) 2002-03-27 EP disclosed
WO-2000066112-A1 CXCR-4 RECEPTOR ANTAGONISTS - THROMBOPOIETIN MIMETICS SMITHKLINE BEECHAM CORPORATION (US) 2000-11-09 WO disclosed