SCHEMBL7477252

SCHEMBL7477252

CCS(=O)(=O)Nc1cccc(C(c2c(O)cc(C(CC3CC3)CC3CCCOC3)oc2=O)C2CC2)c1

nearest known ligand 0.33

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.32
REN P00797 3/20 0.31
MAP1LC3B Q9GZQ8 1/20 0.31
MAP1LC3A Q9H492 1/20 0.31
CYP3A4 P08684 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7482086 0.89 GAA (0.35) BRD4MAP1LC3BMAP1LC3ACYP3A4
SCHEMBL6174348 0.84 MAPK1 (0.34) RENCYP3A4
SCHEMBL7400236 0.82 TRIM24 (0.39)
SCHEMBL7397144 0.81 PDE4B (0.40) BRD4CYP3A4
SCHEMBL6174251 0.81 CYP2C9 (0.38) RENCYP3A4
SCHEMBL7487811 0.80 ADRB3 (0.33) MAP1LC3BMAP1LC3A
SCHEMBL6174752 0.79 NQO1 (0.35) RENCYP3A4
SCHEMBL7405143 0.79 HSD17B2 (0.39) BRD4
SCHEMBL7396533 0.79 KDM4E (0.41)
SCHEMBL7400178 0.79 KCNK3 (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0668860-B1 PYRAN-2-ONES AND 5,6-DIHYDROPYRAN-2-ONES USEFUL FOR TREATING HIV AND OTHER RETROVIRUSES UPJOHN CO (US) 2002-09-11 EP claimed