SCHEMBL7477322

SCHEMBL7477322

CSc1cnc(OCCOc2ncnc(NS(=O)(=O)c3ccc(C(C)(C)C)cc3)c2-c2scc3ccccc23)nc1

nearest known ligand 0.72

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
EDNRB P24530 2/20 0.54
EDNRA P25101 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7480255 0.84 EDNRB (0.63) EDNRBEDNRA
SCHEMBL7477422 0.83 EDNRB (0.58) EDNRBEDNRA
SCHEMBL795873 0.83 EDNRB (0.54) EDNRBEDNRA
SCHEMBL7481169 0.82 EDNRB (0.68) EDNRBEDNRA
SCHEMBL7487690 0.81 EDNRB (0.61) EDNRBEDNRA
SCHEMBL8801730 0.81 EDNRB (0.81) EDNRBEDNRA
SCHEMBL8660604 0.81 EDNRB (0.57) EDNRBEDNRA
SCHEMBL7489110 0.80 EDNRB (0.58) EDNRBEDNRA
SCHEMBL8657549 0.80 EDNRB (0.80) EDNRBEDNRA
SCHEMBL8801001 0.80 EDNRB (0.71) EDNRBEDNRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0959072-B1 Sulfonamide derivative and process for preparing the same TANABE SEIYAKU CO (JP) 2002-09-25 EP claimed
EP-0959072-B1 Sulfonamide derivative and process for preparing the same TANABE SEIYAKU CO (JP) 2002-09-25 EP disclosed
EP-0959072-A1 Sulfonamide derivative and process for preparing the same TANABE SEIYAKU CO., LTD. (JP) 1999-11-24 EP disclosed
US-5739333-A 4-SULFONAMIDO-6-ARYLOXY OR -AMINOALKYLENEOXY,-AMINO, OR -THIOPYRIMIDINES; ENDOLTHELIN ANTAGONISTS; HYPOTENSIVE AND ULCER AGENTS; ASTHMA; RAYNAUD DISEASE; CARDIOVASCULAR DISORDERS TANABE SEIYAKU CO., LTD. (JP) 1998-04-14 US disclosed
EP-0743307-A1 Sulfonamide derivative and process for preparing the same TANABE SEIYAKU CO., LTD. (JP) 1996-11-20 EP disclosed