SCHEMBL7478957

SCHEMBL7478957

COc1cc2nccc(Oc3ccc(NC(=O)Nc4ccc(N)cc4Cl)cc3)c2cc1OC

nearest known ligand 0.84

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
KDR P35968 20/20 0.84
PDGFRA P16234 18/20 0.84

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7481445 0.91 KDR (1.00) KDRPDGFRA
SCHEMBL5204147 0.90 KDR (0.84) KDRPDGFRA
SCHEMBL7485268 0.90 PDGFRA (0.85) KDRPDGFRA
SCHEMBL6864391 0.90 KDR (0.83) KDRPDGFRA
Hydrochloric Acid SCHEMBL5202398 0.90 KDR (0.82) KDRPDGFRA
SCHEMBL3848338 0.89 KDR (0.86) KDRPDGFRA
SCHEMBL7490363 0.88 KDR (0.83) KDRPDGFRA
SCHEMBL27081475 0.87 PDGFRA (0.95) KDRPDGFRA
SCHEMBL29973354 0.87 PDGFRA (0.95) KDRPDGFRA
SCHEMBL7484072 0.87 KDR (0.81) KDRPDGFRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0860433-B1 QUINOLINE DERIVATIVES AND QUINAZOLINE DERIVATIVES INHIBITING AUTOPHOSPHORYLATION OF GROWTH FACTOR RECEPTOR ORIGINATING IN PLATELET AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME KIRIN BREWERY (JP) 2002-07-03 EP disclosed
US-6143764-A ETHER DERIVATIVES OF QUINOLINE, ANTITUMOR AGENTS KIRIN BEER KABUSHIKI KAISHA (JP) 2000-11-07 US disclosed