SCHEMBL7478959

SCHEMBL7478959

C[C@@H](O)[C@@](O)(Cn1cncn1)c1ccc(F)cc1F

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 17/20 0.70
CYP2C9 P11712 11/20 0.70
CYP2C19 P33261 11/20 0.70
LMNA P02545 2/20 0.70
CYP2B6 P20813 1/20 0.70
CYP3A5 P20815 1/20 0.70
CYP3A7 P24462 1/20 0.70
MAPK1 P28482 1/20 0.70
CYP3A43 Q9HB55 1/20 0.70
CYP46A1 Q9Y6A2 1/20 0.70
HSP90AA1 P07900 1/20 0.69
CYP19A1 P11511 1/20 0.69
CYP11B1 P15538 1/20 0.69
CYP11B2 P19099 1/20 0.69
ADRA1A P35348 1/20 0.69
CYP51A1 Q16850 1/20 0.69
CYP1A2 P05177 6/20 0.64
CYP2D6 P10635 6/20 0.64
KCNH2 Q12809 3/20 0.59
ABCG2 Q9UNQ0 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2566503 1.00 CYP3A4 (0.70) CYP3A4CYP2C9CYP2C19LMNACYP2B6
SCHEMBL30485092 1.00 CYP3A4 (0.70) CYP3A4CYP2C9CYP2C19LMNACYP2B6
SCHEMBL1824105 1.00 CYP3A4 (0.70) CYP3A4CYP2C9CYP2C19LMNACYP2B6
SCHEMBL7537507 1.00 CYP3A4 (0.70) CYP3A4CYP2C9CYP2C19LMNACYP2B6
SCHEMBL18717940 1.00 CYP3A4 (0.70) CYP3A4CYP2C9CYP2C19LMNACYP2B6
SCHEMBL2912761 1.00 CYP3A4 (0.70) CYP3A4CYP2C9CYP2C19LMNACYP2B6
SCHEMBL10597737 1.00 CYP3A4 (0.70) CYP3A4CYP2C9CYP2C19LMNACYP2B6
SCHEMBL29357899 0.93 CYP3A4 (0.63) CYP3A4CYP2C9CYP2C19LMNACYP2B6
SCHEMBL28847757 0.93 CYP3A4 (0.63) CYP3A4CYP2C9CYP2C19LMNACYP2B6
SCHEMBL28847754 0.93 CYP3A4 (0.63) CYP3A4CYP2C9CYP2C19LMNACYP2B6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1475370-B1 OPTICALLY ACTIVE AZOLE DERIVATIVE AND PROCESS FOR PRODUCING THE SAME MITSUI CHEMICALS INC (JP) 2009-08-05 EP disclosed
US-7271185-B2 Optically active azole derivative and process for producing the same MITSUI CHEMICALS, INC. (JP) 2007-09-18 US disclosed
US-7271185-B2 Optically active azole derivative and process for producing the same MITSUI CHEMICALS, INC. (JP) 2007-09-18 US disclosed
EP-1071640-B1 ASYMMETRIC SYNTHESIS OF 2-ARYL-1-SUBSTITUTED BUTAN-2,3-DIOLS NAEJA PHARMACEUTICAL INC (CA) 2002-03-13 EP disclosed
EP-1071640-A1 ASYMMETRIC SYNTHESIS OF 2-ARYL-1-SUBSTITUTED BUTAN-2,3-DIOLS Naeja Pharmaceutical Inc. (CA) 2001-01-31 EP disclosed
US-6133485-A Asymmetric synthesis of 2-(2,4-difluorophenyl)-1-heterocycl-1-yl butan-2,3-diols SYNPHAR LABORATORIES, INC. (CA) 2000-10-17 US disclosed
WO-1999052840-A1 ASYMMETRIC SYNTHESIS OF 2-ARYL-1-SUBSTITUTED BUTAN-2,3-DIOLS NAEJA PHARMACEUTICAL INC. (US) 1999-10-21 WO disclosed
EP-0728752-A1 Triazole compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-08-28 EP disclosed
US-5405861-A Fungicides TAKEDA CHEMICAL INDUSTRIES, CO., LTD. (JP) 1995-04-11 US disclosed
EP-0421210-A2 Triazole compounds, their production and use Takeda Chemical Industries, Ltd. (JP) 1991-04-10 EP disclosed